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N-(2-methyl-5-sulfamoylphenyl)-4-(1,3-thiazol-2-yl)piperazine-1-carboxamide
2-(2-chloro-4-fluorophenyl)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-3-(piperidin-3-yl)benzamide
(3R,4R)-1-(2-amino-4-methylpyrimidine-5-carbonyl)-3,4-dimethylpyrrolidin-3-ol
6-fluoro-2-{[methyl(thian-4-yl)amino]methyl}quinolin-4-ol
7-(cyclopropylmethyl)-2-[2-(methylsulfanyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
1-(4-methoxyphenyl)-6,6-dimethyl-4-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]piperazin-2-one
N3-ethyl-N5-[(3-fluorophenyl)methyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
5-ethyl-5-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
3-{[1-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
4-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenyl)-2-methylbutan-2-ol
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[1-(3-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
(1S,5R)-3-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(3-{3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
2-[3-(methoxymethyl)-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(5-methylfuran-2-yl)methyl]acetamide
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-cyclobutanecarbonylpiperidine
5-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-2-methoxyphenol
methyl (2S,4S)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxylate
8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-fluoro-N,2-dimethylbenzamide
N-(2,2-dimethyloxan-4-yl)-N,1-dimethyl-1H-imidazole-2-carboxamide
(1S,5R)-6-[2-(4-fluorophenoxy)ethyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1,3-dimethyl-N-[(1R,3S)-3-[4-(propan-2-yl)piperazine-1-carbonyl]cyclopentyl]-1H-pyrazole-4-carboxamide
N-cyclopentyl-5-[(4-hydroxyphenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-{2-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}imidazolidine-2,4-dione
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2,2-dimethylpropanamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
(2R,3R)-3-amino-1'-(2-methylpyrimidin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N,2-dimethyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-phenyl-1-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}piperidine-4-carbonitrile
3-acetamido-N-[2-(2-ethoxyphenoxy)ethyl]-N-methylbenzamide
1-[4-(4-methoxyphenyl)butanoyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
4-methyl-3-oxo-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-3,4-dihydroquinoxaline-2-carboxamide
(3R)-1-[1-(6-chloro-1,3-benzothiazol-2-yl)piperidin-4-yl]pyrrolidin-3-ol
5-{1-[2-(4-chlorophenyl)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
2-(diethylamino)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
1-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(4-ethylpiperazin-1-yl)ethan-1-one
N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-[1-(pyridin-2-yl)propyl]acetamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
(2S)-2-amino-1-{6-methyl-5-[5-(piperidin-1-ylmethyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}propan-1-one
ethyl 4-{[(3S,4R)-4-ethoxyoxolan-3-yl]amino}piperidine-1-carboxylate
5-(dimethylamino)-2-[(4-methoxypyridin-2-yl)methyl]-2,3-dihydropyridazin-3-one
3-{[1-(dimethyl-1,3-thiazol-4-yl)ethyl]sulfamoyl}-N,N-dimethylbenzamide
[(3R,4R)-1-(6-cyclopropylpyrimidin-4-yl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
1-(4-fluorophenyl)-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
4-[3-(methoxymethyl)pyrrolidin-1-yl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-oxopentanamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide