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N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-methoxyphenoxy)acetamide
1'-(5,6-dimethylpyrimidin-4-yl)-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)propanamide
N-(oxan-4-yl)-1-(3-phenylpropyl)azepan-3-amine
4-{1-[(4-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-1H-indazole-3-carboxamide
3-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}pyridine
N-methyl-N-(2-{[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethyl)methanesulfonamide
1-[(1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
6-(2-fluorophenyl)-N-(2-methoxyethyl)-N-(propan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3S,4S)-4-{ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}-1-(4-methoxybenzoyl)pyrrolidin-3-ol
2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1-(morpholin-4-yl)ethan-1-one
1-(1,3-oxazole-5-carbonyl)-4-(9H-purin-6-yl)-1,4-diazepan-6-ol
[(2-methoxynaphthalen-1-yl)methyl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
7-chloro-2-methyl-4-[4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carbonyl]quinoline
(1,3-benzothiazol-2-ylmethyl)(methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
N-benzyl-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
4-methyl-1-[3-(piperidine-1-carbonyl)benzenesulfonyl]-1,4-diazepan-5-one
1-[1-(4-fluorobenzoyl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-[3-(dimethylamino)propyl]-9-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-1-(propan-2-yl)piperidine
ethyl({[5-(methoxymethyl)furan-2-yl]methyl})({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amine
8-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}quinoline
N,N-dimethyl-1-(2-methyl-1-benzofuran-5-carbonyl)azepan-4-amine
(4aS,8aR)-6-methanesulfonyl-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[(2-chlorophenyl)methyl]-7-fluoro-3-({[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)pyridine-3-carboxamide
2-({[(2-ethoxyphenyl)methyl](ethyl)amino}methyl)benzoic acid
{3-[(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl)methyl]phenyl}methanol
5-oxo-1-[2-(pyridin-2-ylsulfanyl)ethyl]pyrrolidine-3-carboxylic acid
2-{1-benzyl-4-[(3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(pyridin-3-ylmethyl)-4-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)pyrrolidin-2-one
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-3,4,5-trimethoxybenzamide
1-(cyclohexyloxy)-3-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]propan-2-ol
1-ethyl-8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-2-[3-(4-phenoxybenzoyl)piperidin-1-yl]acetamide
8-ethoxy-5-(quinolin-7-ylmethyl)-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
methyl 5-[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)carbamoyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylate
3-methoxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(1-methylpiperidin-4-yl)oxy]-N-(propan-2-yl)benzamide
methyl (2S)-5-(4-acetyl-4-phenylpiperidin-1-yl)-2-amino-5-oxopentanoate
(2-{2-[1-(1H-indole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-butyl-N-ethyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
2-[4-(2-ethylbutyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-[(2-fluorophenyl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-(6-chloro-1,3-benzothiazol-2-yl)piperidin-4-amine
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanol