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3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-[2-(ethylsulfanyl)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
2-(2,3-dihydro-1H-indol-1-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
5-phenyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1,2,3-thiadiazole-5-carboxamide
(3aS,6aS)-5-[(6-methylpyridin-2-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4,6-dimethylpyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N4-{3-[ethyl(methyl)amino]butyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(4aR,7aS)-1-(2-hydroxyethyl)-4-[4-(morpholin-4-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-chloro-2-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-N-(2-methoxyethyl)quinazolin-4-amine
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-(pyrazin-2-yl)propanamide
1-cyclopentyl-4-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-2-one
3-[1-(5-acetylthiophene-3-carbonyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
N-butyl-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-(furan-2-ylmethyl)butanamide
1-phenyl-N-{[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-3-yl]methyl}methanesulfonamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1H-pyrazole-3-carboxamide
3-[(dimethylamino)methyl]-1-[2-(2,3-dimethylphenoxy)ethyl]piperidin-3-ol
2-[3-(4-chlorophenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-6-carboxylic acid
2-(azepan-1-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxoacetamide
3-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}sulfonyl)pyridine
2-{[3-(3-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)-1H-pyrazol-1-yl]methyl}pyridine
1-ethyl-4-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-3-methylpiperazin-2-one
1-methyl-2-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-{1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidine-3-carbonyl}pyridine
4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1-methyl-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-chloro-1,3-dimethyl-4-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N3-ethyl-N1-(3-methylcinnolin-5-yl)pyrrolidine-1,3-dicarboxamide
ethyl 2-({5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}(methyl)amino)acetate
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
3-(4-methyl-1H-pyrazol-5-yl)-1-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}piperidine
(3R)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
N-[2-({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]-N-methylmethanesulfonamide
1-(2-phenylethyl)-8-propyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-cyclopropyl-N-(1-hydroxy-2-methylpropan-2-yl)-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
N,N-dimethyl-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
1-(cyclopropylmethyl)-5-[(4-methoxyphenyl)methyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{4-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-4-oxobutyl}acetamide
1-cyclopropyl-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
methyl 4-[(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)methyl]benzoate
5-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-dimethyl-1H-pyrazole
2-(4-methoxyphenyl)-6-methyl-5-[(4-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-benzyl-5-[(furan-2-ylmethyl)amino]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)ethan-1-one
N-({5-[(2,3-difluoro-4-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
4-(furan-2-ylmethyl)-3-(3-hydroxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
2-(3-fluorophenoxymethyl)-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,3-oxazole-4-carboxamide