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1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-[3-(1H-imidazol-1-yl)propyl]-1-[3-(piperidin-1-ylmethyl)phenyl]urea
N-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)-3,5-dimethoxybenzamide
2-{1-benzyl-4-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-({2-[3-(2-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
(1S,6R)-3-(4-ethenylbenzoyl)-3,9-diazabicyclo[4.2.1]nonane
N-[2-(azepan-1-yl)ethyl]-5-fluoro-N-methylquinazolin-4-amine
N-[1-({[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl)carbamoyl}methyl)-1H-pyrazol-4-yl]-2H-1,3-benzodioxole-5-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl]({[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl})(oxolan-2-ylmethyl)amine
N-[3-(4-chlorophenoxy)propyl]-N,1-dimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
7-cyclohexyl-2-(4-hydroxy-3-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidine
1'-[2-(ethylamino)pyrimidine-5-carbonyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
methyl 6-[(diethylamino)methyl]-3-[2-(3-methylphenyl)acetamido]thieno[2,3-b]pyridine-2-carboxylate
methyl 2-[7-(1-hydroxy-2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]benzoate
N-[1-(4-{[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]furan-3-carboxamide
8-(5-chloropyridin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
3-{2-amino-4-methyl-6-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrimidin-5-yl}propanoic acid
1-ethyl-4-{[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
5-hydroxy-N,1,2-trimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-indole-3-carboxamide
N-[1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-2-phenylethyl]-N-methylthiophene-3-carboxamide
2-({[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
4-{2-[1-(cyclopropanesulfonyl)piperidin-2-yl]ethyl}phenol
N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-2-(pyridin-4-yl)quinoline-4-carboxamide
N-cyclopentyl-N-({4-[(2-fluorophenyl)methoxy]phenyl}methyl)cyclopropanecarboxamide
N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-cyclopropyl-1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-4-phenyl-1H-imidazole
5-(3-{1-[3-(piperidin-1-yl)propyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-methylpiperidin-2-one
(but-2-yn-1-yl)({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(furan-2-ylmethyl)amine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[1-(pyridin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N,5,7-trimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
3-[4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-3,5-dimethyl-1H-pyrazol-1-yl]-1λ6-thiolane-1,1-dione
5-(2-carbamoylethyl)-N-cyclopentyl-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-(2,2-dimethylpropyl)piperazin-2-one
N-[3-(3,4-dimethylphenoxy)propyl]-N-methylpiperidine-4-carboxamide
1-(5-chlorothiophene-2-carbonyl)-3-(1H-imidazol-2-yl)piperidine
4-methyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(4H-1,2,4-triazol-4-yl)pyridine
6-methyl-3-{2-oxa-7-azaspiro[4.5]decane-7-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N-[(3-fluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-1,8-naphthyridine-2-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(furan-2-yl)benzoyl]pyrrolidin-3-yl]methanol
N-[(4-methoxyphenyl)methyl]-1-methyl-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-(pyrimidin-2-yl)piperidin-4-amine
5-[1-(4-methylbenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-[5-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
4-[(3S,4S)-1-(benzenesulfonyl)-4-hydroxypyrrolidin-3-yl]-1,4-diazepane-1-carbaldehyde