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N-ethyl-7,8-dimethyl-2-(2-methylpyrimidin-5-yl)-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
(3S,4R)-3-ethyl-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-methylpiperidin-4-ol
N-(pyrimidin-4-ylmethyl)-1-benzofuran-5-carboxamide
2-(benzyloxy)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
[(3S,5R)-5-[(dimethylamino)methyl]-1-{[3-(morpholin-4-yl)phenyl]methyl}piperidin-3-yl]methanol
8-methoxy-2-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}quinoline
N-ethyl-1-methyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{1-[(4-fluoro-2-methylphenyl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
(isoquinolin-5-ylmethyl)[(4-methanesulfonylphenyl)methyl]methylamine
4-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]-5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidine
5-[5-(2-benzyl-1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-3-amine
2-(4-{[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl}-1,2,3,6-tetrahydropyridin-1-yl)acetamide
2-[(6-ethyl-2-oxo-2H-chromen-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(azepane-1-carbonyl)-N-ethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(cyclopropylmethyl)-5-[2-(3,4-dimethoxyphenyl)acetyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-ethoxyacetamide
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-3-(pyrazin-2-yl)propanamide
4-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 3-acetamido-5-{[4-(1H-indol-3-yl)butan-2-yl]amino}-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N5-cyclooctyl-N3-(cyclopropylmethyl)-4-oxo-N3-propyl-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]morpholine
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-({[(trimethylpyrazin-2-yl)methyl]amino}methyl)pyrrolidin-2-yl]methanol
N-methyl-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
2-[4-(1-methoxyethyl)phenyl]-N,N,5-trimethylpyrimidin-4-amine
N-{2-[(1R,7S)-6-(4-fluoropiperidine-1-carbonyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]ethyl}acetamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[3-(methylsulfanyl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
9-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-({[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})amino}methyl)pyrimidin-2-amine
3-propyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
5-(2,6-difluorophenoxymethyl)-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazole
5-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{[cycloheptyl(pyridin-3-ylmethyl)amino]methyl}-4H-chromen-4-one
4-methyl-2-phenyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazine
2-(2H-1,3-benzodioxol-5-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
4-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-(pyridin-3-yl)morpholine
1-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,4-diazepane-6-carboxylic acid
(1-tert-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)(3-chlorophenyl)methanol
4-(piperazine-1-carbonyl)-N-(pyridin-4-ylmethyl)benzene-1-sulfonamide
1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carboxamide
5-(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
1-benzyl-5-[(cyclopropylmethyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,5R)-1-(1-methylpiperidin-4-yl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
methyl 3-{[1-(cyclohexylmethyl)-3-(dimethylcarbamoyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
4-(4-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}piperazin-1-yl)quinoline
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(5-methoxyfuran-2-carbonyl)pyrrolidine-3-carboxylic acid
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(pyridin-2-yl)ethyl]amino}methyl)piperidin-2-one
N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
6-[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]pyridine-2-carboxylic acid