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N-[(5-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
2-{4-[3-(cyclopentylcarbamoyl)propanoyl]piperazin-1-yl}pyridine-3-carboxamide
7-fluoro-4-methyl-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
7-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butanoic acid
(1S,9S)-11-{6-[(dimethylamino)methyl]-2-methylpyrimidin-4-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
8-[(3,4-dimethylphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[2-(difluoromethoxy)phenyl]methyl}-3-methoxy-1,2-dihydropyridin-2-one
1-[(2-aminopyridin-3-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
1-(carbamoylmethyl)-N-[(2-chloropyridin-3-yl)methyl]-N-methylpiperidine-4-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-{[4-(methylsulfanyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
ethyl 5-(1H-indole-2-carbonyl)-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-{2-[4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]ethyl}aniline
3-[(3R,4S)-4-(dimethylamino)-1-[1-(3-methoxyphenyl)piperidin-4-yl]piperidin-3-yl]propanoic acid
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(thiophen-3-yl)propanamide
(3aR,7aS)-5-methyl-2-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-(pyridin-3-ylmethyl)-4-[4-({2-[2-(trifluoromethyl)phenyl]ethyl}amino)piperidin-1-yl]benzamide
N-(2,3-dihydro-1H-inden-2-yl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-(methoxymethyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)furan-2-carboxamide
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(thiophen-2-ylmethyl)acetamide
1-(4-aminoazepan-1-yl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
methyl 9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-3-(3-methylthiophene-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-{4-[4-({imidazo[1,2-a]pyridin-3-ylmethyl}amino)piperidin-1-yl]phenyl}benzenesulfonamide
3-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-(1-methyl-1H-imidazol-2-yl)pyridazine
N-[(3R,4S)-1-(2-hydroxyethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]-2-(2-oxopiperidin-1-yl)acetamide
4-(5-fluoropyridin-2-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl 4-(2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)butanoate
N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
ethyl 1-[(3-acetylphenyl)carbamoyl]-3-benzylpiperidine-3-carboxylate
2,4-dimethyl-N-(1-{4-[(oxan-4-ylmethyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)benzamide
(4aR,6R,8aS)-2-[(4-chlorophenyl)methyl]-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
N-[(2-fluorophenyl)methyl]-2-({[4-(pyrrolidine-1-carbonyl)phenyl]methyl}amino)acetamide
(2S,4S)-4-amino-1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperazine-1-sulfonamide
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
(3aR,6aR)-2-methyl-5-[6-(morpholin-4-yl)pyrimidin-4-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-acetamido-N-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}pyrrolidine-1-carboxamide
4-benzyl-1-(2,4-dimethylbenzoyl)-3-ethyl-1,4-diazepan-5-one
1-{1-[(8-methylquinolin-5-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
5-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-ethyl-1,2,4-oxadiazole
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[3-(morpholin-4-yl)propyl]amine
7-(2,3-dimethoxyphenyl)-9-methoxy-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4,6-dimethyl-1-(2-oxo-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
(3R,5S)-N3-(4-fluorophenyl)-N5-(oxolan-2-ylmethyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
1'-(2-methyl-1,3-thiazole-4-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-6-methoxypyrimidin-4-amine
3-{5-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
5-(2,4-dimethoxyphenyl)-N-[3-(methylsulfanyl)propyl]-1,2,4-triazin-3-amine