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2-{1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-2-yl}pyridine
1-[(2-fluorophenyl)methyl]-4-(2-methyloxane-2-carbonyl)-1,4-diazepane
methyl 5-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-5-oxopentanoate
methyl 1-[(3R,5S)-1-(2-ethylbutyl)-5-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[(2,3-difluoro-6-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane
1'-(1,7-dimethyl-1H-indole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-4-yl)ethyl]amine
3-(3,4-difluorophenyl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
methyl (2S,4S)-4-(furan-2-amido)-1-(propan-2-yl)pyrrolidine-2-carboxylate
N-cyclohexyl-3-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
(4aS,7aR)-N-tert-butyl-4-[(4-ethylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-(2-ethoxyphenyl)-3-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}urea
1-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-2-phenylethan-1-one
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
(1S,5R)-6-(1-methyl-1H-pyrazole-3-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
(4S)-3,3,4-trimethyl-1-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]piperidin-4-ol
1-(4-methoxyphenyl)-6,6-dimethyl-N-(oxan-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(2-methoxyacetyl)-N-[(5-methylpyrazin-2-yl)methyl]piperidine-4-carboxamide
N,5-dimethyl-3-phenyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-4-carboxamide
methyl 2-[1-(tert-butylcarbamoyl)propyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
N-[5-(4-methyl-1H-pyrazol-1-yl)pyridin-2-yl]acetamide
methyl 3-{[4-(methoxycarbonyl)phenyl]methyl}-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
ethyl 4-[4-(2-methylpropyl)-3-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl]piperidine-1-carboxylate
N-cyclopropyl-3-(4-hydroxyphenyl)-N-(pyridin-3-ylmethyl)benzamide
2-benzyl-9-(cyclobutylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(1H-indol-2-yl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
ethyl 5-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-1-(3-chlorophenyl)-1H-pyrazole-4-carboxylate
1-(2-acetamidoacetyl)-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-methyl-1H-indazole-3-carboxamide
5-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-4-methylpyrimidin-2-amine
N-methyl-1-(2-methylpropyl)-5-oxo-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrrolidine-3-carboxamide
4-({4-[2-(dimethylamino)ethoxy]phenyl}methyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1,2,5-thiadiazole-3-carboxamide
6-({4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,1,6-trimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
1-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
3-[3-(ethoxymethyl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1-methylpiperidine
2-cyclopropyl-9-[(4-methyl-1H-imidazol-5-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-{1-methyl-5-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
5-(1-benzothiophen-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-1-[(3-methylphenyl)methyl]azepan-2-one
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]ethan-1-ol
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
N2,N2-dimethyl-N4-[(3-methyl-1-benzofuran-2-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
6-[2-fluoro-6-(propan-2-yloxy)phenyl]pyridin-3-amine
1-[(4-methyl-5-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-ol
2-[(3R,4S)-3-(2-cyclobutylacetamido)-4-phenylpyrrolidin-1-yl]-N-methylacetamide
4-(naphthalen-2-ylmethyl)-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[5-(methoxymethyl)furan-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-3-(2-methoxyphenyl)propanamide
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide