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2-{4-[(2,5-difluorophenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-(4-ethylpiperazin-1-yl)-3-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
1-(4-benzylpiperazin-1-yl)-3-[1-(3-methoxybenzoyl)piperidin-3-yl]propan-1-one
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]benzamide
(3S,4R)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
3-[(4-{1,9-dioxaspiro[5.5]undecan-4-yl}piperazin-1-yl)methyl]benzonitrile
2-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-3,4-dihydroquinazolin-4-one
1-benzyl-N,N-dimethyl-5-[2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(adamantan-1-ylmethyl)({[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
2-(4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}morpholin-3-yl)-N-[(2-fluorophenyl)methyl]acetamide
2-tert-butyl-4-hydroxy-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrimidine-5-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[(3-methylpyridin-4-yl)methyl]amine
[1-(cyclopent-1-ene-1-carbonyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
2-{4-[(5-ethylfuran-2-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
methyl (2S,4R)-4-[4-(1H-pyrazol-1-yl)benzamido]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-4-propylpyrimidine
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-5-methyl-1,3-oxazole-4-carboxamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}oxane-4-carboxamide
(4aR,8aR)-2-(4-cyclopentylpyrimidin-2-yl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
8-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(1-{1-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-cyclopropyl-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-methylpyrrolidine-2-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(morpholin-4-yl)acetamide
2-(4-ethylpiperazin-1-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}acetamide
3-[5-(2,4,5-trimethylphenyl)-1,2,4-oxadiazol-3-yl]pyridazine
1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
N-cyclopropyl-2-{[1-(1-hydroxypropan-2-yl)piperidin-4-yl]oxy}-4-methoxybenzamide
4-(2,2-diphenylethyl)-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
1-[(1S,5R)-6-(3-chlorobenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-{4-[(4-methyl-3-phenylpiperazin-1-yl)methyl]thiophen-2-yl}ethan-1-one
1-[4-ethoxy-3-(trifluoromethyl)phenyl]-5-oxopyrrolidine-3-carboxylic acid
(3R,4R)-4-amino-1-({3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-5-yl}methyl)piperidin-3-ol
N-(1-{7-[(2-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
5-(4-{[(1,3-benzoxazol-2-yl)amino]methyl}piperidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
3-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
4-(1H-imidazol-4-ylmethyl)-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(5S,9aS,9bS)-5-(2,6-difluorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
methyl 4-{[(2S,4R)-2-[(diphenylmethyl)carbamoyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidin-1-yl]methyl}benzoate
8-(1-benzofuran-5-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 9-[3-(dimethylamino)propoxy]-3-(4-fluorobenzoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-methyl-1-[2-(morpholin-4-yl)ethyl]-5-phenylpiperidin-2-one
(2S,4R)-N-(2,3-dihydro-1H-inden-2-yl)-4-(2,5-dimethylfuran-3-amido)-N-methylpyrrolidine-2-carboxamide
3-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
(2S)-1-{[3-(4-cyclopentyl-6-oxo-1,6-dihydropyrimidin-2-yl)phenyl]methyl}-N-ethylpyrrolidine-2-carboxamide
1-cyclopentanecarbonyl-N-[2-(3-methylpyridin-2-yl)ethyl]piperidine-4-carboxamide
9-(2-fluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-({1-[(2,4-difluoro-3-methoxyphenyl)methyl]piperidin-3-yl}methyl)morpholine