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4-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}-2-phenylpyrimidine
ethyl 1-(1-{1,3-dioxo-2-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carbonyl)piperidine-3-carboxylate
2-[3-(1-phenyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-1,2,3-triazol-4-yl)acetamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[(4-fluoro-3-methoxyphenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-3-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
1-[({[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}carbamoyl)methyl]piperidine-4-carboxamide
1'-(2-amino-5,6-dimethylpyrimidin-4-yl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N4-[2-(1-benzylpyrrolidin-3-yl)ethyl]-6-methylpyrimidine-2,4-diamine
1-(3,4-dimethylphenyl)-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(pyridin-3-yl)acetamide
5-[benzyl(methyl)amino]-2-[(3R)-3-hydroxy-3-phenylpropyl]-2,3-dihydropyridazin-3-one
5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-2,4-dimethyl-1,3-thiazole
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-pyrazol-5-yl)benzamide
1-(1-benzylpiperidin-4-yl)-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
1-[2-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-2-oxoethyl]-3-methyl-1,2-dihydroquinoxalin-2-one
4-[2-(3-methoxyphenoxy)ethyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-1H-pyrrole-2-carboxamide
8-[(2-ethylpyrimidin-4-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{1-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]ethyl}pyrimidine
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-phenoxyethyl)piperazine
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-hydroxy-N-methyl-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-4-(pyridin-3-yl)piperazine-1-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]acetamide
N-(5-fluoro-2-methylphenyl)-3-{[(2S)-5-oxopyrrolidin-2-yl]formamido}propanamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(pyrrolidin-3-yl)benzamide
1-{[(2S,4S)-4-fluoro-1-(1,3,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]methyl}-3,3-dimethylurea
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(1-methylpiperidin-2-yl)ethyl]acetamide
5-({[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]carbamoyl}amino)-2-methoxy-N-methylbenzamide
3-[({5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}amino)methyl]-6-cyclopentyl-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[3-(1H-pyrazol-1-yl)propyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
1,3-dimethyl-2,6-dioxo-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-methyl-4-(4-{8-methyl-2,8-diazaspiro[4.5]decane-2-carbonyl}phenyl)butan-2-ol
N-ethyl-4-methyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl){[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-[(3-hydroxypropyl)sulfamoyl]benzamide
2-{[7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}acetamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-methanesulfonylpropan-1-one
2-{4-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
methyl 3-(furan-2-amido)-5-({[4-(2-hydroxyethoxy)phenyl]methyl}amino)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2,2-dimethyl-N-{1-[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
methyl[(3-{2-[1-(3-methylthiophene-2-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](quinolin-8-ylmethyl)amine
N-[(3-fluorophenyl)methyl]-2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]acetamide
1-(5-hydroxypyrazine-2-carbonyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
(3R,4R)-4-methyl-1-(1-phenylcyclopropanecarbonyl)-3-(propan-2-yl)pyrrolidin-3-ol
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
[(2S,4R,5R)-5-(4-chlorophenyl)-4-({[(3,4-dimethoxyphenyl)methyl]amino}methyl)-1-ethyl-2-methylpyrrolidin-2-yl]methanol
N-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-1H-indazole-3-carboxamide
4-benzyl-3-{1-[(1R,2S)-2-propylcyclopropanecarbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-cyanocyclopropane-1-carboxamide