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8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-N-propyl-2,8-diazaspiro[5.5]undecane-2-carboxamide
3-{[3-(dimethyl-1,2-oxazol-4-yl)propyl]sulfamoyl}-N,N-dimethylbenzamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(pyrimidin-2-yl)pyrrolidin-3-yl]methanol
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)pyridine-3-carboxamide
3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1H-indazole
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-(2-ethylphenyl)-2-oxo-2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]acetamide
2-(3-{1-[2-(1-methylpiperidin-2-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
N-(1-methyl-3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}-1H-pyrazol-5-yl)acetamide
methyl N-(1-oxo-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-2-yl)carbamate
2-butoxy-1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrimidin-4-amine
N,N,4-trimethyl-3-[(pentylcarbamoyl)methyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
methyl 2-{3-[(4-cyclohexylpiperazin-1-yl)methyl]-7-methyl-2-oxo-1,2-dihydroquinolin-1-yl}acetate
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-ethylphenyl)methyl]-N-methylacetamide
1-(cyclohexylmethyl)-4-{[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}pyrrolidin-2-one
(2S,4S)-4-amino-N-ethyl-1-(5-oxo-5-phenylpentanoyl)pyrrolidine-2-carboxamide
methyl 8-{[3-(benzyloxy)phenyl]methyl}-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
5-(azocane-1-carbonyl)-1-cyclopentylpiperidin-2-one
N,1-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-indole-6-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-cyclohexylbenzamide
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-3-fluoro-N-(oxolan-2-ylmethyl)benzamide
1-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-indole-3-carboxamide
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-[(3,4-difluorophenyl)methyl]-2-[(4-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
methyl 5-({[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}amino)-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(ethylamino)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]pyrimidine-5-carboxamide
N-{1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methyl-1-oxopropan-2-yl}thiophene-2-carboxamide
N-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]methanesulfonamide
1-{4-[({[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}amino)methyl]phenyl}pyrrolidin-2-one
2-(2-phenylethyl)-4-(propane-2-sulfonyl)morpholine
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N,N,4-trimethyl-3-{[methyl(pentyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-fluoro-6-methyl-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
2-oxo-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-2,3-dihydro-1H-imidazole-4-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}propanamide
N-(2-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-[2-(5-methylfuran-2-yl)phenyl]urea
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]pyridin-2-amine
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1,1-dioxo-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1λ6-thiane-4-carboxamide
methyl 1-cyclohexyl-2-oxo-3-[2-(4H-1,2,4-triazol-4-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(oxan-4-yl)piperazine
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylate
(4S)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
4-(1,3-benzothiazol-2-yl)-2-({benzyl[2-(dimethylamino)ethyl]amino}methyl)phenol
3-(3-chloro-2-fluorophenyl)-1-(1-cyclopropanecarbonylpiperidin-3-yl)urea
2-({4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperazin-1-yl}methyl)benzonitrile