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4-(5-fluoro-2-methylphenyl)-3-[(propan-2-yloxy)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,5-difluorophenyl)-2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}acetic acid
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylacetamide
1-(2-methanesulfonylethyl)-4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperazine
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidine-3-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-3-{[(5-methylfuran-2-yl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
(3E)-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}hex-3-en-1-one
N-(5-chloro-2-methoxyphenyl)-3-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]propanamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(2-fluoro-5-methylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
3-{2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2,6,6-trimethyl-1-propyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-[2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethoxy]ethan-1-ol
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2-(2-phenyl-1,3-thiazol-4-yl)-N-(pyridin-4-ylmethyl)acetamide
ethyl 1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
N-[1-(4-chlorophenyl)ethyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3,3-dimethylurea
1-(cyclopent-3-en-1-yl)-5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazole
3-{2-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-2,5-dione
2-(pent-4-enoyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
(3aS,6aS)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-octahydropyrrolo[2,3-c]pyrrole
4-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(3-phenylpropyl)morpholine
[4-methyl-5-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methanol
1-methyl-2-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine-1-carbonyl}azepane
6-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridin-3-ol
2-(4-{[(2-methoxyethyl)(methyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-6,7-dimethyl-1H-1,3-benzodiazole
3-({1-cyclohexyl-3-hydroxy-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
N,N-dimethyl-4-(4-methylpent-3-en-1-yl)benzamide
2-(4-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}morpholin-3-yl)acetic acid
4-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}thiomorpholine
6,6-dimethyl-1-(4-methylphenyl)-N-(oxan-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-[2-({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-(2-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
N-[1-(4-chlorophenyl)cyclopropyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
5-(2,6-dimethylphenoxymethyl)-N-[(2-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
5-chloro-3-methyl-N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-1H-indole-2-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
2-[5-(2-methyl-1,3-benzothiazol-5-yl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-[2-(2-methoxyphenoxy)phenyl]-6-oxa-9-azaspiro[4.5]decane-9-carboxamide
2-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}benzoic acid
4-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]benzonitrile
5-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-3-(1-phenylcyclopropanecarbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{5-[1-(4-phenyl-1H-imidazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
N-(isoquinolin-5-ylmethyl)-N-methyl-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-[({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[2-(2,5-dimethoxyphenyl)acetyl]-1-methylpiperazine-2-carboxylic acid
8-(1H-indol-2-ylmethyl)-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione