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2-(1H-indol-3-yl)-1-(4-{2-[(4-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)ethan-1-one
5-{[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2,5-dimethyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(1S,5R)-6-[(2,4-difluorophenyl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
[(1-cyclopentylpiperidin-4-yl)methyl][(1-methyl-1H-imidazol-2-yl)methyl](pyridin-3-ylmethyl)amine
1-cyclopropanecarbonyl-2-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]piperidine
8-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}quinoline
(2S)-2-amino-1-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-imidazol-4-yl)propan-1-one
1-(5-methoxy-2-{[methyl(2-phenoxyethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
3-[2-(4-acetyl-1,4-diazepan-1-yl)-2-oxoethyl]-4-[(2-methylphenyl)methyl]piperazin-2-one
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N-[2-(dimethylamino)ethyl]-N-methylpiperidin-3-amine
1-[3-methoxy-5-(trifluoromethyl)phenyl]-3-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-methylurea
(4aS,7aR)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-6,6-dioxo-N-(propan-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[1-(2,2-dimethylbutanoyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
6-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
8-(3-chloro-4-fluorobenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-{6-hydroxy-4-[4-(hydroxymethyl)benzoyl]-1,4-diazepan-1-yl}acetic acid
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(2-ethyl-1H-1,3-benzodiazol-1-yl)propan-1-one
(4S,4aS,8aS)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
ethyl 4-[4-(4-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
2-amino-6-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1-(2-methoxyethyl)pyrrolidin-2-one
1-[(5-chlorothiophen-2-yl)methyl]-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)quinoline
7-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[(1S)-1-phenylethyl]-1H-1,3-benzodiazole-5-carboxamide
3-(3,4-dimethoxyphenyl)-1-[4-(pyrimidin-4-yl)piperidin-1-yl]propan-1-one
N-(3,4-difluorophenyl)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})(thiophen-3-ylmethyl)amine
N-[2-(1H-indol-3-yl)ethyl]-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
7-(1,3-benzothiazol-2-yl)-4-(1H-1,2,4-triazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(1-propyl-1H-imidazol-2-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-phenylprop-2-ynamide
2-{4-[(2-chlorophenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[(3R)-3-hydroxypyrrolidin-1-yl]-3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]propan-1-one
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(pyridin-4-yl)propanamide
2-(dimethyl-1,2-oxazol-4-yl)-N-{[7-(pyridin-3-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}acetamide
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-[2-(methylsulfanyl)benzoyl]piperidine
ethyl 4-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-1H-pyrazole-3-carboxylate
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-cyclopropanecarbonyl-2-(3-fluoro-4-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-[4-(2-hydroxyethyl)piperidin-1-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(4-methyl-1,3-oxazol-5-yl)-1H-1,2,4-triazol-3-yl]acetamide
2-[2-(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
5-cyclopropanecarbonyl-1'-[(2S)-1-ethylpyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-4-(3-methyl-1-benzothiophen-2-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyrazin-2-yl)-1,4-diazepan-5-one
N-{[5-methyl-2-(4-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}pyridine-2-carboxamide