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4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-N,N-dimethyl-4-oxobutanamide
(2R,3R)-3-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(2R,3R)-2-ethoxy-1'-(3-fluoro-4-methoxybenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-benzyl-3-[2-(2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-1-methyl-2,3-dihydro-1H-indol-2-one
4-[(4-methylphenyl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1,4-diazepan-5-one
1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
6-(methoxymethyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,3R)-3-amino-N-{2-[4-(dimethylamino)phenyl]ethyl}cyclopentane-1-carboxamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-ol
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-[(5-{[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}pyrimidin-2-yl)amino]acetic acid
2-(5-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]sulfonyl}thiophen-2-yl)pyridine
1-{6-[2-(4-chlorophenyl)morpholin-4-yl]pyrimidin-4-yl}piperidin-4-ol
[7-(3-chloropyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
7-[(2-methoxyphenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-{4-[1-(pyridin-3-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}pyridine
(2R,6R)-4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3,6-dimethyl-N-[2-(N-methylmethanesulfonamido)ethyl]-1-benzofuran-2-carboxamide
2-cyano-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]benzamide
6-methoxy-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}hexan-1-one
1-[4-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenyl]ethan-1-one
5-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(3-methoxyphenyl)propanamide
N-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-methyl-2-(3-methylphenoxy)propanamide
1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-phenylpiperidin-4-yl]ethan-1-one
5-acetyl-N-methyl-N-[2-(4-methylpiperidin-1-yl)ethyl]thiophene-3-carboxamide
1-(2,4-dimethylphenoxy)-3-[(oxan-4-yl)amino]propan-2-ol
N-[phenyl(pyridin-4-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide
1-(5-methoxy-2-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
3-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1-{4-[2-(pyrrolidin-1-yl)ethyl]phenyl}urea
(3R,4R)-1-(3,6-dimethylpyrazin-2-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
ethyl 1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
1-(3-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
N-(2-methoxyethyl)-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-cyclopropyl-1-{1-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-(1H-1,2,3-benzotriazol-5-yl)-1-cyclohexyl-1-(pyridin-2-ylmethyl)urea
4-[4-(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]phenol
(1R,5S,6S)-N-(2,3-dihydro-1H-inden-2-yl)-3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
5-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
2-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-4H-chromen-4-one
9-(5-methylpyrazine-2-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-[(3-chloro-5-fluorophenyl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-ethyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(4-chlorophenyl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
5-chloro-1,3-dimethyl-4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}sulfonyl)-1H-pyrazole
6-methoxy-3-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1-benzofuran-2-carboxamide