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2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
2-phenyl-N-{1-[1-(pyridine-3-sulfonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
2-(dimethylamino)-4-methyl-N-(2-oxoazepan-3-yl)pyrimidine-5-carboxamide
N-(2-methoxyethyl)-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}benzene-1-sulfonamide
2-(2-methoxyethyl)-9-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(carbamoylmethyl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)piperidine-4-carboxamide
3-methyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
5-(hydroxymethyl)-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}furan-2-carboxamide
1-({4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}methyl)-1H-imidazole
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}pent-4-enamide
3-methyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
2-{[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-5-[(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylformamido)methyl]benzoate
1-benzyl-4-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}piperazine
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-cyclopentylpiperidin-2-one
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
4-(3-fluoropyridin-4-yl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-(oxolan-2-ylmethyl)acetamide
N-[(4-chlorophenyl)(pyridin-3-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
5-methyl-1'-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{5-[2-(2-methoxyethyl)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}propanoic acid
1-({3-[1-(dimethylamino)ethyl]phenyl}methyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-[3-(1H-indol-2-yl)phenyl]-1-(propan-2-yl)piperidine-3-carboxamide
2-{1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-yl}benzoic acid
1-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(1H-indol-1-yl)ethyl]-N-methylpropanamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-[(5-ethylpyridin-2-yl)methyl]-1-(3-hydroxyphenyl)-N-methyl-5-oxopyrrolidine-3-carboxamide
N-(4-cyanophenyl)-3-(3-phenylpropanoyl)piperidine-1-carboxamide
N-[(2-ethylpyrimidin-5-yl)methyl]-1-[(2-fluorophenyl)methyl]-N-methylpiperidin-3-amine
methyl 3-[3-(2-methoxyphenyl)propanoyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-{[1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)pyrrolidin-3-yl]methyl}benzoic acid
4-(3-benzyl-1H-pyrazol-5-yl)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine
N,N-diethyl-1-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidine-3-carboxamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[2-(4-fluorophenyl)morpholin-4-yl]acetamide
3-(3-methoxybenzoyl)-1-[(5-methylfuran-2-yl)methyl]piperidine
N-(3-methylphenyl)-3-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidin-4-yl}propanamide
1-(piperidin-1-yl)-3-[2-(pyrrolidin-1-ylmethyl)phenoxy]propan-2-ol
2-[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(4-methylpyrimidin-2-yl)piperidin-4-ol
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-(2-methoxy-2-methylpropyl)acetamide
4-(4-methoxyphenyl)-6-(pyridazine-3-carbonyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
(3R,4R)-4-amino-1-({3-[3-(trifluoromethyl)phenoxy]phenyl}methyl)piperidin-3-ol
9-(3-methylbut-2-enoyl)-1,4,9-triazaspiro[5.5]undecan-5-one
2-cyclopropyl-8-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
4-{[2-(diethylamino)-2-(furan-2-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid