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methyl 3-[(3-methoxyphenyl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-benzothiazole-6-carboxamide
1'-(3,4-difluorobenzoyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[(2,3-dimethoxyphenyl)methyl]-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
1-[2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]-3,3-dimethylurea
N-[(3S,7S,8aS)-3-(cyclohexylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
(4-{[4-(3,5-dichloro-2-methoxyphenyl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methanol
1-{1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}azepane
(3S,7S)-5-[4-(hydroxymethyl)benzoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-{2-[({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]phenoxy}ethan-1-ol
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[3-(1H-1,2,4-triazol-1-yl)propyl]cyclopentane-1,3-dicarboxamide
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(1-methylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
1-(2-methoxyphenyl)-N-methyl-N-(quinoxalin-6-ylmethyl)-1H-pyrazole-4-carboxamide
3-[(4-ethylphenyl)methyl]-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-5-(3-methoxyphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
[(1-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
N-[3-(4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}piperidin-1-yl)phenyl]pyridine-3-carboxamide
4-[4-(4,4-difluoropiperidin-1-yl)piperidin-1-yl]-6-ethyl-N,N-dimethylpyrimidin-2-amine
1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(2S)-1-(2-ethylpyrimidine-5-carbonyl)pyrrolidine-2-carbonyl]morpholine
1-({2-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]phenyl}methyl)pyrrolidin-2-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
3-methyl-1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
N-(3-{4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]piperidin-1-yl}phenyl)pyridine-3-carboxamide
1-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-(4-methylphenyl)acetamide
1-(2,5-dichlorophenyl)-3-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}urea
N-(1-{1-[4-(4-hydroxyphenyl)butan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(oxolan-3-yl)propanamide
4-({5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)morpholine
3-[1-(cyclopent-3-ene-1-carbonyl)piperidin-3-yl]-N-[(3,4-difluorophenyl)methyl]propanamide
2-[2-(ethoxymethyl)-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-amine
(1R,2S,9R)-11-(quinoxaline-5-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)acetamide
2-[5-(4-cyanophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
3-[1-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetyl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(5-ethyl-2-methylpyrimidin-4-yl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
N-[(1-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)methyl]furan-2-carboxamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-[1-(pyridin-2-yl)propan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-[3-(2-ethylpiperidine-1-carbonyl)piperidin-1-yl]-2-[2-(3-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
(2-methoxyethyl)[(4-methylphenyl)methyl](pyridin-4-ylmethyl)amine
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(1H-imidazole-4-carbonyl)piperidine
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,5S)-1-[(2-fluoro-5-methoxyphenyl)methyl]-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
2-methyl-5-(propan-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
(3R,4S)-1-[3,5-bis(trifluoromethyl)benzoyl]-4-cyclopropylpyrrolidin-3-amine
2-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one