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3-methyl-5-{[(4-methyl-1,3-thiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazole
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-propyl-1H-pyrazole-5-carboxamide
(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-{[(2-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
5-phenyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1,2-oxazole-3-carbonyl)piperidin-3-yl]propanamide
1-(3-{[bis(prop-2-en-1-yl)amino]methyl}phenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(furan-3-ylmethyl)acetamide
2-methyl-4-[4-({4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}methyl)phenyl]butan-2-ol
1-ethyl-5-[1-(2-methylpropanoyl)piperidine-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[(2-fluorophenyl)formamido]-N-(naphthalen-1-ylmethyl)propanamide
6-[2-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]-2,3-dihydropyridazin-3-one
(3aR,6aR)-2-[2-(benzyloxy)ethyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylnaphthalene-2-carboxamide
2-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
1-methyl-4-[(5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}furan-2-yl)methyl]piperazine
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-2-(pyrrolidin-3-yl)benzamide
1-(cyclopentylmethyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
N-benzyl-N-(cyclohexylmethyl)-2-[methyl(piperidin-4-yl)amino]acetamide
5-ethyl-2-methyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine
1-cyclohexyl-4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(5-{[4-(cyclopentyloxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
2-hydroxy-N-(4-methoxy-3-pentanamidophenyl)pyridine-3-carboxamide
methyl 4-{[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]amino}butanoate
9-(2-methoxyethyl)-1-methyl-4-(pyrazin-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[2-(morpholin-4-ylmethyl)phenyl]-1-[2-(pyridin-2-yl)ethyl]urea
1-(2-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}ethyl)imidazolidin-2-one
2-cyclopropyl-1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
6-methyl-N-[2-(5-methylthiophen-2-yl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-4-(morpholin-4-yl)butan-1-one
6-[(3-methoxyphenyl)methoxy]-4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-1-(2-methylpropyl)-1,4-diazepan-2-one
1,5-dimethyl-3-[3-(2-methylphenyl)piperidine-1-carbonyl]-1H-indazole
1-(1'-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
N-{[1-(6-cyclopropylpyrimidin-4-yl)piperidin-4-yl]methyl}acetamide
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-(3-phenyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[(4-chloro-3-fluorophenyl)methyl](methyl)(oxan-4-ylmethyl)amine
[2-(4-{[4-(propan-2-yloxy)phenyl]methyl}piperazin-1-yl)pyridin-4-yl]methanol
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[1-(pyridin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
6-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
5-(3-fluorophenoxymethyl)-N-(isoquinolin-5-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
methyl 5-(3-methylthiophene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-[4-(3-methoxypropyl)piperidin-1-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
1-(cyclopropylmethyl)-6-{[(3-methoxyphenyl)methyl](methyl)amino}-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
methyl 4-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)piperazine-1-carboxylate
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]benzonitrile