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1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[5-(2,6-dimethoxyphenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-[(5-methylpyrazin-2-yl)methyl]-8-[3-(methylsulfanyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[(1-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
(1R,2S)-N1-(prop-2-en-1-yl)-N2-[(2,4,6-trimethylphenyl)methyl]cyclohexane-1,2-dicarboxamide
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
1-ethyl-4-({4-[(3-fluorophenyl)methoxy]-3-methoxyphenyl}methyl)piperazin-2-one
2-({1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}methyl)benzonitrile
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]amine
1-(dimethyl-1,3-thiazol-2-yl)-5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
2-(2H-1,2,3-benzotriazol-2-yl)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)acetamide
5-(2,4-difluorophenoxymethyl)-N-methyl-N-(thiophen-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-[3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
1-(2-{[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]amino}pyrimidin-4-yl)piperidin-4-ol
2-phenoxy-1-{4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-1-yl}ethan-1-one
1-(2-methoxyphenyl)-4-(1-phenylcyclopropanecarbonyl)piperazin-2-one
3-butyl-4-(3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-ethyl-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]urea
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
(1S,5R)-3-{[3-(2-hydroxyethoxy)phenyl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{5-[1-(2-phenyl-1H-imidazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
N-[1-({[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
1-(3-cyanophenyl)-3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
4-({[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}methyl)benzoic acid
3-methoxy-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpropanamide
(2S)-2-{2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}propanamide
N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-imidazol-4-yl)propan-1-one
1-methyl-2-oxo-8-[3-(pyridin-3-yl)propanoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
7-{2-[4-ethyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]ethyl}-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
3-methyl-8-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(3-chloro-4-hydroxyphenyl)ethan-1-one
N-[2-(methylsulfanyl)ethyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(4-methyl-1,3-thiazole-5-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(1-{[3-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)pyridine
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)[1-(pyridin-4-yl)ethyl]amine
1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(3-acetylphenoxymethyl)-N-(2-hydroxyethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
2-chloro-N-{[1-(quinoxaline-5-carbonyl)piperidin-3-yl]methyl}benzamide
1-[(3-hydroxy-4-methoxyphenyl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
N5-(2-ethyl-1H-1,3-benzodiazol-6-yl)-N2-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2,5-dicarboxamide
4-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
4-methoxy-1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperidine
5-cyclopropanecarbonyl-1'-[(3,4-difluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 3-benzyl-1-(2,4-dimethoxybenzenesulfonyl)piperidine-3-carboxylate