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N-[(3,4-dimethoxyphenyl)methyl]-2,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-indole-7-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-{2-[(dimethylcarbamoyl)amino]acetyl}pyrrolidine-3-carboxylic acid
7-(2-methoxyethyl)-2-(5-propylthiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-({5-[(N-methylmethanesulfonamido)methyl]-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
1-{2-[1-cyclohexyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidin-2-yl)methanol
{1-[(4-methyloxan-4-yl)methyl]piperidin-4-yl}(thiophen-2-yl)methanol
3-[1-(azepane-4-carbonyl)piperidin-4-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-[3-(3-methylphenoxy)propyl]acetamide
methyl 1-(2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperidine-4-carboxylate
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
3-methyl-4-(2-methyl-4-phenylpyridine-3-carbonyl)-1-(2-methylpropyl)piperazin-2-one
2-[5-(2H-1,3-benzodioxol-5-yl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
N-cyclopentyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]benzamide
4-ethyl-3-{[1-(1H-indol-2-ylmethyl)piperidin-4-yl]methyl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(cyclohexylmethyl)-4-(oxane-4-carbonyl)morpholine
7-(2-hydroxyethyl)-2-({7-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4S)-4-amino-1-(4-chloro-2-methylbenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
1-[(3-chloro-4,5-diethoxyphenyl)methyl]-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
N-[4-(4-{methyl[2-(oxan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
N-(1-hydroxybutan-2-yl)-4-(1H-indol-3-yl)-N-(pyridin-3-ylmethyl)butanamide
2-(butylsulfanyl)-6-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]pyrimidin-4-amine
N-[3-chloro-4-(2,2-dimethylpropanamido)phenyl]-5-methylpyrazine-2-carboxamide
1-[(2-chlorophenyl)methyl]-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-cyclopentanecarbonyl-4-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]piperidine
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-1-cyclohexyl-1H-1,2,3-triazole-4-carboxamide
3-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-9-methoxy-N-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl}-1,3-benzoxazole
(3S,4S)-4-[({5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)methyl]piperidin-3-ol
(4-{[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-phenyl-1H-imidazol-1-yl]methyl}oxan-4-yl)methanol
4-{[4-(2-{1-[2-(thiophen-3-yl)acetyl]piperidin-2-yl}ethoxy)phenyl]methyl}piperazine-1-carbaldehyde
2-{1'-[(2-methyl-1,3-oxazol-4-yl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl]methanol
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidine-4-carboxylic acid
3-(2-oxoazepan-1-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]propanamide
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1,2,5-thiadiazole-3-carboxamide
7-{[ethyl(4-hydroxybutyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-fluorophenyl)-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
5-acetyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}thiophene-3-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(naphthalen-2-ylmethyl)piperidine
1-[2-({[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
1-methyl-3-(propan-2-yl)-N-(thiolan-3-yl)-1H-pyrazole-5-carboxamide
N-(cyclopent-3-en-1-yl)-2-{4-[(2r,4r)-6,8-dioxo-5,7-diazaspiro[3.4]octane-2-carbonyl]morpholin-3-yl}acetamide
1-cyclohexyl-4-(5-methoxyfuran-2-carbonyl)-1,4-diazepane
N,6-diethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2,6-dimethoxypyridine-3-carbonyl)piperidine-3-carboxylate