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5-(4-cyclohexylphenyl)-3-[3-(methoxymethyl)piperidin-1-yl]-1,2,4-triazine
1-[(4-chloro-3-fluorophenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-{[4-(aminomethyl)phenyl]methyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-(butan-2-yl)-6-cyano-N-(3-phenylprop-2-yn-1-yl)pyridine-3-carboxamide
5-phenyl-2-(pyridin-4-yl)-4-[1-(thiophen-2-ylmethyl)piperidin-3-yl]pyrimidine
9-[(3-chlorophenyl)methyl]-3-oxa-9-azaspiro[5.5]undecane
2-[1'-(2,4-dimethylpyrimidine-5-carbonyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
3-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
3-(3-fluorophenyl)-3-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
(2S)-1-acetyl-N-{[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyrrolidine-2-carboxamide
3-{5-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
4-{[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amino}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
4-[(4-{[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]morpholine
3-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
2,5-dimethyl-4-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
4-(3,5-difluoro-4-methoxyphenyl)-1-[2-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole
3-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-1-ethyl-7-methyl-1,4-dihydro-1,8-naphthyridin-4-one
1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-(2,4-dioxoimidazolidin-1-yl)-N-methylbenzamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{spiro[indene-1,4'-piperidine]-1'-yl}butan-1-one
2-[4-({[(4-methoxyphenyl)carbamoyl]amino}methyl)-1,2,3,6-tetrahydropyridin-1-yl]acetamide
N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-1H-indole-5-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(2,4-difluorophenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[2-(2-fluorophenyl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
1-(2-hydroxyacetyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
4-{[1-(2,2-dimethylbutanoyl)pyrrolidin-3-yl]methyl}benzoic acid
2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-2-[4-(pyridin-4-yl)piperidin-1-yl]acetic acid
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-4-(piperidin-3-yl)benzamide
N-(3-chloro-4-methylphenyl)-8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
4-ethyl-3-{2-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
N-(2-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
N-{[(3S,4S)-1-(5-ethylthiophene-2-carbonyl)-3-hydroxypiperidin-4-yl]methyl}-2,2-dimethylpropanamide
methyl (1R,3S,3aR,6aS)-3-(4,5-dimethylthiophen-2-yl)-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-methyl-2-(pyridin-4-yl)-N-[1-(pyrimidin-4-yl)ethyl]quinoline-4-carboxamide
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
N-benzyl-1-(2-hydroxyethyl)-5-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-methyl-2-phenyl-N-[2-(1H-1,2,4-triazol-1-yl)propyl]pyrimidin-4-amine
2-{2-[4-phenyl-5-(2,4,5-trifluorophenyl)-1H-imidazol-1-yl]ethoxy}ethan-1-ol
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(2,4-dioxo-1,3-diazinan-1-yl)benzamide
1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
1-methyl-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
(3aR,6aR)-2-acetyl-5-(1,3-thiazol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-2-(1-methyl-1H-imidazol-2-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]benzamide
2-{4-[(4-chlorophenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N-methyl-5-(oxolan-2-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}thiophene-2-carboxamide
(1R,7S)-3-tert-butyl-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(2R)-1-({4-[(1-ethyl-4-methyl-1H-pyrazol-5-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxamide