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9-[(4-fluoro-3-methylphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-methoxy-3-methylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(5,6-dimethylpyrimidin-4-yl)piperidine-4-carboxylic acid
N-{[1-(1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
(3S,4S)-4-(morpholin-4-yl)-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidin-3-ol
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-6-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-(2-methoxypyridin-3-yl)benzamide
N-[(3-fluorophenyl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
(1R,3S)-3-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}cyclopentan-1-amine
2-hydroxy-N-methyl-4-(methylsulfanyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-[2-(methylsulfanyl)benzoyl]piperidine
6-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-(pyridin-3-ylmethyl)urea
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
4-[(3-ethyl-1H-pyrazol-5-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-one
2-phenyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-5-carboxamide
3-cyclopentyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]propanamide
2-[methyl(quinolin-5-ylmethyl)amino]-N-[4-(N-methylacetamido)phenyl]acetamide
1-phenyl-N-[(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)methyl]methanesulfonamide
4-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)butan-1-ol
2-(4-methylphenyl)-5-{4-[(pyrimidin-2-yl)amino]piperidine-1-carbonyl}pyrimidin-4-ol
2-(4-hydroxyphenyl)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}acetamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1,4-diazepan-5-one
1-(3-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)ethan-1-one
N-[2-(2-ethoxyethoxy)phenyl]-4-(pyridin-4-yl)piperazine-1-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
5-[(4-fluoro-3-methoxyphenyl)methyl]-3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-[3-({[3-(pyrrolidin-1-yl)propyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(3R,4R)-1-{[5-(4-chlorophenyl)furan-2-yl]methyl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(thiophen-2-yl)butanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopentylimidazo[1,2-a]pyridine-6-carboxamide
N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N4-[2-(1H-imidazol-4-yl)ethyl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
2-methanesulfonyl-5-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-1-(3-methoxypropyl)-1H-imidazole
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[benzyl(methyl)amino]-3-(4-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
(2R)-2-{[2-(4-tert-butylphenoxymethyl)-4-hydroxypyrimidin-5-yl]formamido}propanamide
2-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]-N-phenylacetamide
1-(pyridin-3-ylmethyl)-4-[3-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3-azaspiro[5.5]undecan-9-amine
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-3-(3-methoxyphenyl)propanamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
5-(3,4-dimethoxyphenyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,4-triazin-3-amine
1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
6-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]pyridine-2-carboxylic acid
7-(3-chlorophenyl)-4-(2-ethoxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[3-(oxan-4-yl)-5-[5-(oxolan-2-yl)thiophen-2-yl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-(2-{1-[2-(4-methoxyphenoxy)acetyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide