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3-(1H-imidazol-1-ylmethyl)-N-[1-(pyridin-3-ylmethyl)-1H-pyrazol-5-yl]piperidine-1-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(1-benzylpiperidin-3-yl)acetamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
(3S,7S)-5-[3-(pyridin-3-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N2,N2,N4,N4-tetramethyl-7-(pyridine-3-sulfonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-[3-(3-methoxyphenyl)phenyl]-1-(oxan-4-yl)piperidine-4-carboxamide
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
2-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
3-hydroxy-1-(2-methoxyethyl)-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
N-cyclopropyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
N-(1-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
4-[(6-ethyl-2-methylquinolin-4-yl)formamido]-N,4-dimethylpentanamide
1-phenylmethanesulfonyl-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-({4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
(2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-4-[(1H-imidazol-2-ylmethyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
1-methyl-3-{1-[(2S)-oxolan-2-ylmethyl]-4-phenyl-1H-imidazol-5-yl}-1,2-dihydroquinolin-2-one
N-(2-cyclobutyl-7-{4-[hydroxy(thiophen-2-yl)methyl]piperidine-1-carbonyl}-1-methyl-1H-1,3-benzodiazol-5-yl)-2-methoxyacetamide
7-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
ethyl 2-{[2-(4-chlorophenyl)morpholine-4-carbonyl]amino}acetate
5-{[(benzylsulfamoyl)(methyl)amino]methyl}-N-methylpyrimidin-2-amine
(1R,3S)-3-(2-aminoethoxy)-7-(2-chloro-4-fluorobenzoyl)-7-azaspiro[3.5]nonan-1-ol
4-methyl-1-[3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
6-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}pyridine-2-carboxylic acid
(3S,4S)-4-(4-fluorophenyl)-1-[(6-methylquinolin-5-yl)methyl]piperidin-3-ol
3-(2-ethylbutyl)-8-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(4-cyclopentyl-3-oxopiperazine-1-carbonyl)-1,2-dihydroquinoxalin-2-one
1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3-phenylpiperazine
1-[4-methyl-6-(methylamino)pyrimidin-2-yl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-[4-(dimethylamino)phenyl]-N-methylpropanamide
N-[(2R,3R)-2-methoxy-1'-(1,2,5-thiadiazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
1-(2-methylphenyl)-4-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperazin-2-one
5-[(2-fluorophenyl)methyl]-5-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
1-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(5S,9aS,9bS)-5-(furan-2-yl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(difluoromethoxy)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
5-(4-chloro-1-ethyl-1H-pyrazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-({2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)benzoic acid
N,N-dimethyl-7-(piperidine-1-carbonyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-2-(3,4,5-trimethoxyphenyl)acetamide
2-cyclopropyl-4-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidine-5-carboxamide
9-(4-fluoro-3-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[4-(oxan-4-yl)piperazin-1-yl]methyl}pyridin-2-amine
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(pyridin-4-yl)propan-1-one
N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(methylsulfanyl)ethan-1-one
[5-({methyl[(5-methylthiophen-2-yl)methyl]amino}methyl)-2-(propan-2-yloxy)phenyl]methanol
(2S,4R)-1-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-N-ethyl-4-(furan-3-amido)pyrrolidine-2-carboxamide
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}amine
(1R,7S)-6-(morpholine-4-carbonyl)-3-[2-(pyridin-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
6-[(2E)-3-(4-chlorophenyl)prop-2-enoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide