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8-[3-cyclopropyl-5-(1,2,3-thiadiazol-4-yl)-1H-1,2,4-triazol-1-yl]quinoline
ethyl 4-oxo-5-phenoxy-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxylate
N-methyl-5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxamide
1-{[5-(2,1,3-benzoxadiazol-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,3-dimethylurea
[2-(2-chloro-6-methoxyphenyl)pyridin-4-yl]methanol
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
N-(3,3-diphenylpropyl)-6-[(3-ethoxy-2-hydroxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-phenyl-1-[3-(pyridin-4-yl)azetidin-1-yl]butan-1-one
N-benzyl-2-(pyridin-2-yl)pyrrolidine-1-sulfonamide
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)cyclopentanamine
1-(3-{4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl}phenyl)imidazolidin-2-one
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
(3R,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(1H-pyrazol-1-yl)butanamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
2-(3-methoxypropyl)-9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
7-(2-cyclohexylethyl)-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-amino-N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]pyridine-3-carboxamide
3-({1-[5-(methoxymethyl)thiophene-2-carbonyl]pyrrolidin-3-yl}methyl)benzamide
1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-4-hydroxypiperidine-4-carboxylic acid
(4aR,7aS)-4-[(2-fluoro-4-methoxyphenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-(6-chloropyridin-3-yl)-3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-methylurea
2-methyl-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-4-carboxamide
5-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-3-[(2,3-dimethoxyphenyl)methyl]-5-methylimidazolidine-2,4-dione
5-(4-chloro-3-methyl-1H-pyrazol-5-yl)-1-cyclohexyl-3-cyclopropyl-1H-1,2,4-triazole
2-{3-cyclopentyl-5-[2-(methylsulfanyl)pyridin-3-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-(3-hydroxyquinoxalin-2-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,2,3-trimethylquinoxaline-6-carboxamide
9-[2-oxo-2-(piperazin-1-yl)ethyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[(3,5-dimethylphenyl)formamido]ethyl}-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-(thiophen-3-yl)piperidine-1-carboxamide
5-[5-(5-fluoro-1H-indol-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[5-({[3-(4-fluorophenoxy)propyl](methyl)amino}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
1-methyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[1-(3-hydroxy-4-methylbenzoyl)pyrrolidin-3-yl]benzoic acid
1-(benzyloxy)-8-(thiophene-3-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
3-(2H-1,3-benzodioxol-5-yl)-1-(morpholin-4-yl)-3-phenylpropan-1-one
3-[1-(2,5-dimethoxybenzoyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
5-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
[(4-chloro-3-fluorophenyl)methyl]({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(4-methylphenyl)methyl]amine
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(3-ethyl-1,2-oxazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-2-phenyl-N-[1-(1,3-thiazol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
(1R,5R)-3-(pyrimidin-2-yl)-6-(thiophen-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 7-oxo-9-[3-(pyridin-3-yl)propoxy]-3-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-ethanesulfonamido-N-ethyl-1-methyl-N-(oxolan-2-ylmethyl)-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1,2-oxazole-3-carboxamide
4-(5-phenyl-1,2,4-oxadiazol-3-yl)-2-(trifluoromethyl)morpholine
1-{2-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]pyrimidin-4-yl}piperidin-4-ol