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N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
2-(pyridin-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-benzotriazole-5-carboxamide
[2-(2,5-dimethylphenoxy)ethyl](methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
3-[3-({[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(2,3-dimethoxyphenyl)methyl]amine
1'-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]spiro[indene-1,4'-piperidine]
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-2-(2-phenylethyl)piperidine
1-{1-[1-(6-ethoxy-4-methylquinazolin-2-yl)piperidin-4-yl]piperidin-4-yl}-2-methylpropan-1-ol
6-fluoro-N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[2-(pyridin-2-yl)ethyl]quinoline-4-carboxamide
4-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}pyridine
N-[(2-ethoxyphenyl)methyl]-N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
2-(azepan-1-yl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-[5-(2-methyl-1-phenoxypropyl)-1,2,4-oxadiazol-3-yl]pyridazine
1-{3-[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
1-[5-(methoxymethyl)furan-2-carbonyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
[(5-ethylpyridin-2-yl)methyl](furan-2-ylmethyl)(thiophen-3-ylmethyl)amine
methyl[2-methyl-2-(morpholin-4-ylmethyl)propyl](quinolin-5-ylmethyl)amine
[(3R,4R)-1-(4-cyclopentylpyrimidin-2-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-{[4-(cyclohexylamino)quinazolin-2-yl]methyl}piperazine-1-carbaldehyde
methyl 4-({[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazol-4-yl]formamido}methyl)benzoate
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(1,3-oxazol-5-yl)benzamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethylpyrimidine-5-carboxamide
8-[(4-methoxy-3-methylphenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-fluoro-2-{[2-(hydroxymethyl)piperidin-1-yl]methyl}quinolin-4-ol
1-[(1s,4s)-4-aminocyclohexyl]-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(thiomorpholin-4-yl)pyridine-3-carboxamide
2-[(3R,4S)-3-(5-ethylthiophene-3-amido)-4-(propan-2-yl)pyrrolidin-1-yl]acetic acid
4-{[(6-methyl-2-propylpyrimidin-4-yl)amino]methyl}benzene-1-sulfonamide
1-cyclopropyl-N-[3-(2-fluorophenyl)propyl]-5-oxopyrrolidine-3-carboxamide
2-[5-(2-ethyl-1-benzofuran-3-yl)-4-phenyl-1H-imidazol-1-yl]propane-1,3-diol
2-(4-chloro-2-{[2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]methyl}phenoxy)acetamide
2-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-4-enamide
1-(1H-imidazole-4-carbonyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
2-[ethyl({[(3S,4R)-4-(hydroxymethyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
(4aR,8aS)-N,N-dimethyl-1-(2,3,6-trifluorobenzoyl)-decahydro-1,6-naphthyridine-6-sulfonamide
2,5-dimethyl-3-(4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
1-(furan-2-carbonyl)-4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1,4-diazepane
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
4-(pyridin-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidin-2-amine
ethyl 1-(8-methyl-3-{[(thiophen-2-ylmethyl)amino]methyl}quinolin-2-yl)piperidine-4-carboxylate
2-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
4-{5-[(2-ethyl-1-benzofuran-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-methyl-1H-pyrazole
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(methylsulfanyl)pyrimidine
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
N-cyclohexyl-3-[(6-methoxypyrimidin-4-yl)amino]propanamide
ethyl 4-{2-[(2-ethylpiperidin-1-yl)methyl]-8-methylquinazolin-4-yl}piperazine-1-carboxylate