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ethyl({[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(2-methylprop-2-en-1-yl)amine
1-[4-(3-{[(adamantan-1-yl)amino]methyl}-7-(methylsulfanyl)quinolin-2-yl)piperazin-1-yl]ethan-1-one
N-(2-fluorophenyl)-3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
(1R,5R)-6-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-[4-(methylsulfanyl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}pyrrolidin-3-ol
(4aS,7aR)-1-benzoyl-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-2-(4-fluorophenyl)piperidine
2-(dimethylamino)-N,4-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrimidine-5-carboxamide
5-(methoxymethyl)-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
5-cyclopropyl-4-{[4-(3-fluoro-2-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-methyl-1H-pyrazole
2-[(5-acetylthiophen-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(4-fluorophenyl)-4-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]butan-1-one
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
9-{[2-(ethylamino)pyrimidin-5-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-fluoroethyl)-3-{[2-(5-methylthiophen-2-yl)ethyl]sulfamoyl}benzamide
(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)({[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl})amine
1-[3-(difluoromethoxy)benzoyl]-3-(2,6-dimethylphenoxy)azetidine
(1R,3S)-3-amino-N-ethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]cyclohexane-1-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2,2-dimethylbutanamide
N-(butan-2-yl)-1-(4-methoxyphenyl)-N-(pyridin-4-ylmethyl)cyclopropane-1-carboxamide
2-(4-methoxy-3,5-dimethylphenyl)pyridine-4-carboxamide
9-hydroxy-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
3-({4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)pyrrolidin-3-ol
4-(1,4-diazepane-1-sulfonyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]benzamide
3-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-2H-chromen-2-one
4-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
2-methyl-5-[2-(2-{[4-methyl-6-(methylamino)pyrimidin-2-yl]amino}ethyl)morpholin-4-yl]-2,3-dihydropyridazin-3-one
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
N-(1-benzylpiperidin-4-yl)-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(1-acetylpiperidin-4-yl)oxy]-N-(cyclohexylmethyl)-3-methoxybenzamide
N-cyclooctyl-1-(2-methoxyethyl)-4-oxo-5-(4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(4-carbamoylpiperidin-1-yl)-2-[2-fluoro-6-(propan-2-yloxy)phenyl]acetic acid
5-(3-methylbutanoyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
5-acetyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]thiophene-2-carboxamide
2-(furan-2-yl)-5-{1-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]-1H-imidazol-2-yl}pyrimidine
N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1-(oxan-4-yl)piperidine-4-carboxamide
6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-4-(quinoxaline-5-carbonyl)-1,4-diazepan-2-one
2-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-6-methylpyridine-3-carboxylic acid
methyl 2-(2-{[(2-methoxyethyl)(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl)piperidine-1-carboxylate
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
3-methyl-5-{[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,2-oxazole
3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{5-[2-(trifluoromethyl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-[4-(3-ethyl-3-hydroxypiperidine-1-carbonyl)phenoxy]-1-(piperidin-1-yl)ethan-1-one
2-(ethylamino)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}pyrimidine-5-carboxamide
2-(4-fluorophenyl)-4-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}morpholine
N-(2-hydroxy-3-methoxypropyl)-4-(piperazine-1-sulfonyl)benzamide