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N-[(3S,4R)-1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2,3-dihydro-1H-indol-1-yl)ethan-1-one
8-(1,3-benzothiazol-2-ylmethyl)-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N'-(3-ethylphenyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]butanediamide
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]propanamide
4-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
6-[4-(propan-2-yloxy)benzoyl]-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
7-[1-(methoxymethyl)cyclobutanecarbonyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[1-(1,5-dimethyl-1H-indazole-3-carbonyl)piperidin-3-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(3-cyano-4,6-dimethylpyridin-2-yl)phenyl]acetamide
2-methyl-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxamide
1-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}piperidine-4-carboxamide
3-(1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)urea
4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-[(2R)-pyrrolidin-2-ylmethyl]benzamide
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N-(propan-2-yl)-1-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-5-(2,4,5-trimethylphenyl)-1H-imidazole
N-[2-(2-fluorophenyl)-1-[1-(quinoxalin-6-ylmethyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
2-(2,1,3-benzothiadiazol-5-ylmethyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-{[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}-N-(oxolan-2-ylmethyl)benzamide
(5S,9aS,9bS)-5-[(E)-2-(4-methoxyphenyl)ethenyl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-methyl-N-(2-methylprop-2-en-1-yl)-5-propyl-1-benzofuran-2-carboxamide
3-(3,4-difluorophenyl)-5-(3,5-dimethoxybenzoyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(4-benzylpiperazin-1-yl)-3-[1-(3-methylbut-2-en-1-yl)piperidin-3-yl]propan-1-one
(1R,5S,6S,7S)-3-(2-aminoethyl)-6-[1-(3-chlorophenyl)-1H-1,2,4-triazol-5-yl]-10-oxa-3-azatricyclo[5.2.1.01,5]decan-4-one
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(6-methylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-7-methyl-1,2-dihydroquinolin-2-one
1-[(3S,4R)-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
5-(2,6-difluorophenoxymethyl)-N-methyl-N-(2-phenoxyethyl)-1,2-oxazole-3-carboxamide
2-[3-(piperidin-1-ylmethyl)piperidin-1-yl]-4-(pyrrolidine-1-carbonyl)pyridine
1-(1-methyl-1H-pyrrol-2-yl)-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethane-1,2-dione
3-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
8-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[4-(4-{[3-(methylsulfanyl)propyl]amino}piperidin-1-yl)phenyl]-5-phenylpentanamide
1-[(1S,5R)-6-(4-methoxy-2-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]acetamide
5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(1H-1,2,3-benzotriazol-4-yl)-3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethylurea
1-(6-methylpyridin-3-yl)-3-{2-[(trifluoromethyl)sulfanyl]ethyl}urea
4-[(4-fluorophenyl)methanesulfonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[cyclohexyl(methyl)amino]-3-(2-{[methyl(propan-2-yl)amino]methyl}phenoxy)propan-2-ol
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{2-[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]-2-oxoethyl}pyrrolidin-2-one
N-[(3-chlorophenyl)methyl]-3-(1H-pyrazol-1-yl)benzamide
2-(4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
1-ethyl-3-[3-(pyridin-3-yl)propyl]-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}-3-(pyridin-4-yl)propan-1-one
N-[(3R,4R)-1-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide