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2-(3-fluorophenyl)-5-(oxan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(4-chlorophenoxy)-N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]pyridine-3-carboxamide
4-(piperidin-3-yl)-N-[2-(pyrazin-2-yl)ethyl]benzamide
N-cyclopropyl-3-(5-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanamide
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]-6-methyl-4H-pyran-4-one
methyl 3-{[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}benzoate
(2R)-2-(hydroxymethyl)-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}pyrrolidine-1-carboxamide
2-{4-[(2-methoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(4-methoxy-3-methylphenyl)methyl]piperidine
methyl 1-(2-methoxyethyl)-3-(3-phenylpropanamido)-5-({[2-(trifluoromethyl)phenyl]methyl}amino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(3,5-difluorophenyl)methyl]-8-(2-methoxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
1-cyclopropanecarbonyl-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]piperidine-4-carboxamide
4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-1-(propan-2-yl)pyrrolidin-2-one
(3S,9aR)-8-(cyclopropylmethyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(cyclobutylmethyl)-2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-(oxolan-2-ylmethyl)acetamide
3-({7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenol
3-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}-4H-chromen-4-one
[3-({1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
N-(1,3-benzoxazol-2-ylmethyl)-5-(3-methoxyphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
ethyl[2-(morpholin-4-yl)ethyl](quinolin-4-ylmethyl)amine
3-(2-methoxyethyl)-5-[1-(naphthalen-2-yloxy)ethyl]-1,2,4-oxadiazole
N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
2-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
(3aS,7aR)-5-methyl-2-(4-methyl-1H-imidazole-5-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-ethyl-4-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}pyrimidine
3-{5-[1-(1H-pyrazol-1-yl)propyl]-1,2,4-oxadiazol-3-yl}pyridazine
1-(2-methoxy-4-{[methyl(thian-4-yl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4,4-dimethylpiperidine
(1R,3S,5S)-8-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
N-(propan-2-yl)-2-(4-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazin-1-yl)acetamide
1-(3-ethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-phenyl-5-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]pyrimidin-2-amine
3-(4-methyl-1,4-diazepane-1-carbonyl)-N-[(3-methyloxetan-3-yl)methyl]benzene-1-sulfonamide
4-hydroxy-N-[(4-hydroxyphenyl)methyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
2-methyl-4-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylpentanamide
5-methyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
(1R,5S,8S)-8-hydroxy-N-[2-(2-phenoxyethoxy)phenyl]-3-azabicyclo[3.2.1]octane-3-carboxamide
5-[5-chloro-2-(propan-2-yloxy)phenyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
2-{5-cyclopropyl-4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-5-methyl-4-(thiophen-2-yl)pyrimidine
2-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-2-yl]pyridine
2-[3-(2-phenylethyl)-5-[1-(pyrrolidin-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]pyridine
N3-ethyl-N1-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)pyrrolidine-1,3-dicarboxamide
4-(3-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-N-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-(2-{8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[2-(diethylamino)ethyl]-2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-ethylacetamide
N3-cyclooctyl-N5-ethyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[5-(2,4-dimethoxyphenyl)-1-(2-methylphenyl)-1H-1,2,4-triazol-3-yl]acetamide