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5-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-[5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pyridin-2-yl]azepane
N-(3,4-dimethoxyphenyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
2-{4-[(8-fluoroquinolin-2-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-[(5-methylfuran-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
(3R,4R)-1-[(4-chloro-2-fluorophenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-[2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-(3-ethylphenyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carboxamide
4-methoxy-6-[4-(2-methoxyphenoxy)piperidin-1-yl]pyrimidin-2-amine
1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
3-(1-butyl-1H-imidazol-2-yl)-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidine
3-({4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}methyl)benzonitrile
N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(3-phenyl-1H-pyrazol-1-yl)acetamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pentan-3-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(pyridin-2-yl)-8-{[4-(pyridin-2-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(6-methylpyridin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-ol
2-[5-(1-ethyl-1H-pyrazol-3-yl)-4-phenyl-1H-imidazol-1-yl]-N-(1,3-thiazol-2-yl)acetamide
4-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-2-amine
N-(adamantan-2-yl)-5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-(1-{[1-(furan-2-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
methyl 5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-(2H-1,3-benzodioxol-5-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}-1,5-dimethyl-1H-pyrazole
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propane-1-sulfonamide
methyl 1-ethyl-5-({[3-(2-hydroxyethoxy)phenyl]methyl}amino)-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
N-(9H-fluoren-9-yl)-6-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-N-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
2-[4-(pyridin-4-yl)piperazin-1-yl]-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)piperidine
methyl 2-{[5-(4-fluorophenyl)-4-[1-(4,4,4-trifluorobutanoyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N,5-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(2,5-dimethoxyphenyl)-2-[4-(5-oxo-1,4-diazepan-1-yl)piperidin-1-yl]acetic acid
1-cyclopentyl-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
3-(2,5-dimethylfuran-3-yl)-5-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[(3S,4R)-1-[2-(4-fluorophenoxy)acetyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
2-[2-(dimethylamino)ethyl]-8-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[3-(2-ethylphenoxy)azetidin-1-yl]-N,N-dimethylpyrazin-2-amine
N-(thiolan-3-yl)-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
7-methyl-2-[(3-methylthiophen-2-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(2H-1,3-benzodioxol-5-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}acetamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}pyrrolidin-3-yl]methanol
(3aS,6aR)-5-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one