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{5-[(2-chloro-4-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)pyridine-3-carboxamide
2-(5,6-dimethylpyridin-2-yl)benzoic acid
1-methyl-1-[1-(4-methylpyridin-2-yl)propan-2-yl]-3-[3-(methylsulfamoyl)phenyl]urea
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
2-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)morpholin-3-yl]-1-(thiomorpholin-4-yl)ethan-1-one
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
4-(1H-imidazol-1-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}benzamide
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-[(2,4,5-trimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-4-(thiophene-2-carbonyl)piperazine
N-methyl-4-[(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)methyl]benzamide
2-methoxy-1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
(1R,5R)-6-(2,6-difluoro-4-methoxybenzoyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
[(3R,4R)-4-[(dimethylamino)methyl]-1-[2-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methanol
methyl 3-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(1-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
4-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-6-methoxypyrimidin-2-amine
1-(4-{4-[methyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
6-[(diethylamino)methyl]-N-(4-methoxy-2-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[6-(benzylamino)pyridin-3-yl]-5-oxopyrrolidine-3-carboxylic acid
{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}(methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
(2S,4S)-4-amino-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(ethanesulfonyl)-1-(2-methoxyethyl)-5-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-1H-imidazole
(2S,4R)-4-amino-1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-N-methylpyrrolidine-2-carboxamide
2-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
N-[(4-ethoxyphenyl)methyl]-2-(2-hydroxyphenyl)-N-(2-methoxyethyl)acetamide
2-(2-chlorophenyl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-amino-7-(1H-indole-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}acetamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(2-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
{[2-(4-ethylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}({spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl})amine
[(2-fluoro-5-methoxyphenyl)methyl]({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-(cyclopropylmethyl)-7-[1-(propan-2-yl)piperidine-4-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S)-2-{3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamido}propanamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[(5-methyl-1H-indol-3-yl)methyl]amine
2-methanesulfonamido-N-[(3R,4S)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
N-(3-cyclopentylpropyl)-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-methoxy-1-[1'-(4-methyl-1,3-thiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-(6-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridin-3-yl)ethan-1-one
N-[2-(2-methoxyphenyl)ethyl]-2-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}quinazolin-4-amine
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
1-[2-(dimethylamino)-4-(4-hydroxypiperidin-1-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-2-propoxyethan-1-one
5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-(oxolan-3-yl)-1-phenyl-1H-1,2,4-triazole
2-methoxy-5-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyrimidine
1-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
3-{4-[4-(pyridin-4-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-2H-indazole