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1'-{[4-(pyridin-3-yl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide
2-{4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}propanamide
1-[(2-chlorophenyl)methyl]-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
4-(4-phenyl-1-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-imidazol-5-yl)pyridine
11-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-4-(3-hydroxypropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(2,3-dimethoxyphenyl)methyl]-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carboxamide
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
4-[5-cyclopropyl-4-(morpholine-4-carbonyl)-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
4-[4-(8-methoxyquinolin-2-yl)piperazin-1-yl]quinazoline
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
3-{1-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]piperidin-4-yl}propanamide
2-[4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)morpholin-2-yl]ethan-1-amine
N-[2-(3-methoxyphenyl)phenyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
1-[1'-(2-hydroxypyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-({1-[(3-chloro-4-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-2-cyclopropylacetamide
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
(3R,5S)-1-[(3-chlorophenyl)methyl]-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-[(4-methoxy-2,3-dimethylphenyl)methyl]pyrrolidin-3-amine
N-cyclopentyl-N'-[(2-phenylphenyl)methyl]butanediamide
(4aS,7aR)-1-(cyclopropylmethyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-methylpiperidine
1-(2-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazine
4-{[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]methyl}benzonitrile
(1R,2S,9R)-11-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-(1H-pyrazol-1-yl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]butan-1-one
N4,N4,5-trimethyl-N2-[3-(pyrrolidin-1-yl)propyl]pyrimidine-2,4-diamine
4-methoxy-2-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrimidine
5-[4-(dimethylamino)phenyl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
1-(4-{[8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}thiophen-2-yl)ethan-1-one
[1-ethyl-5-(5-ethyl-1,3,4-oxadiazol-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
methyl 3-benzamido-6-({methyl[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
(4aR,7aS)-1-(2-methoxyacetyl)-4-[3-(pyridin-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S)-1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)pyrrolidin-3-ol
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-3-methylbenzamide
1-(cyclohexylmethyl)-4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
2-{[cycloheptyl(pyridin-3-ylmethyl)amino]methyl}-3-methoxyphenol
methyl 5-[2-(2-methylpropanamido)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(1S,6R)-9-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
1,3-dimethyl-N-[(2S)-oxolan-2-ylmethyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2-{[1-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]sulfanyl}-4,6-dimethylpyrimidine
6-oxo-N-(pyridin-3-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
(5S,9aS,9bS)-5-(2-chloro-4-fluorophenyl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
7-chloro-3-({[1-(furan-2-yl)ethyl]amino}methyl)-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
N-[(3-fluorophenyl)methyl]-4-methyl-5-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine