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N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
1-(4,6-dimethylpyridine-3-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
(1S,5R)-3-(oxan-4-yl)-6-[4-(1H-pyrazol-3-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-cyclopropanecarbonyl-8-[(4-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methoxy-N-(1-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)acetamide
N-benzyl-N-methyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
ethyl 1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-4-(2-methoxyethyl)piperidine-4-carboxylate
(3S,5S,9S)-5-{[(2-methoxyphenyl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
N-[2-(1H-imidazol-4-yl)ethyl]-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(3-methylpiperidine-3-carbonyl)piperidine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(5-methylfuran-2-yl)methyl](pyridin-4-ylmethyl)amine
6-(adamantan-1-ylmethyl)pyrimidin-4-amine
(4aS,7aR)-6,6-dioxo-N-(propan-2-yl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
3-(4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
7-(5-chloropyridin-2-yl)-4-(1-methylpiperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-({4-methyl-5-[1-(2-methylpyrimidin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
5-[1-butyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-1H-pyrrole-3-carbonitrile
8-(2-ethylpyridine-4-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopentyl-N-[3-(1H-indazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
8-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-cyclopropyl-2-methyl-N-[(3-methylthiophen-2-yl)methyl]imidazo[1,2-a]pyrimidine-3-carboxamide
2-(4-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}cyclohexyl)-1H-1,3-benzodiazole
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-4-methoxybenzamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(methylsulfanyl)ethyl]amine
2-{5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}acetic acid
ethyl 4-({4-[1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazine-1-carboxylate
1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
5,6-dimethyl-2-oxo-N-(2-oxoazepan-3-yl)-1,2-dihydropyridine-3-carboxamide
N-({8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-ethyl-5-[6-fluoro-4-(thiomorpholine-4-carbonyl)quinolin-2-yl]pyrimidin-2-amine
6-[(4-fluorophenyl)methoxy]-4-(furan-3-carbonyl)-1-(propan-2-yl)-1,4-diazepan-2-one
2-(5-acetylthiophen-3-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]ethan-1-one
1-{3-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]phenyl}imidazolidin-2-one
N,8-dimethyl-3-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-cyclopropyl-N-[(3-methylthiophen-2-yl)methyl]morpholine-2-carboxamide
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(5-phenyl-1,3,4-thiadiazol-2-yl)-7-azaspiro[3.5]nonan-1-ol
2-methyl-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(thiophen-2-ylformamido)propanamide
1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-ol
(4S)-3-[2-oxo-2-(piperazin-1-yl)ethyl]-4-phenyl-1,3-oxazolidin-2-one
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,3-benzodiazole-2-carboxamide
N-[1-(4-methylpyridin-2-yl)propyl]-1,4-dithiepan-6-amine
(4S)-1-[1-(furan-2-ylmethyl)piperidin-4-yl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
3-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-N-ethylbenzamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-[2-(cyclopent-1-ene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-2-(2-fluorophenyl)acetamide
2-({benzyl[(1R,2R)-2-hydroxycyclohexyl]amino}methyl)pyridine-3-carboxylic acid
4-(3-methyl-1H-pyrazol-1-yl)-2-(1,2-oxazol-5-yl)phenol
3-{[1-(2,3-dihydro-1H-inden-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione