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1,3-dimethyl-6-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
[(3R,4S)-1-[(3-fluoro-2-methylphenyl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
3-{2-[5-(3-fluoro-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
N-(2-methylpropyl)-2-{3-[3-(2-methylpyrimidin-4-yl)phenyl]-1H-pyrazol-1-yl}acetamide
2-[(3R,4S)-3-(butane-1-sulfonamido)-4-cyclopropylpyrrolidin-1-yl]acetamide
N-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
N-cyclopentyl-4-[4-(2-methoxyphenyl)piperidin-1-yl]-4-oxobutanamide
(2S,4S,5R)-4-{[2-(dimethylamino)ethyl](methyl)carbamoyl}-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[(2S)-pyrrolidin-2-ylmethyl]benzamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
methyl 3-(2-methoxyacetamido)-5-{[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]amino}-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-phenylpiperidine-1-carboxamide
3-[1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]propan-1-ol
2-(5-oxopyrrolidin-2-yl)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
(2S)-2-amino-2-cyclohexyl-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-[2-(ethylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
1-[2-(furan-2-yl)azepan-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
4-[(4-hydroxyquinolin-2-yl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}cyclopropanecarboxamide
(1R,3S)-7-[1-(thiophene-2-carbonyl)piperidin-4-yl]-7-azaspiro[3.5]nonane-1,3-diol
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-ethylpyrimidine-5-carboxamide
2-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}morpholine-2-carboxamide
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
1-(2-methoxyacetyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(1,3-thiazol-2-yl)pyrrolidin-3-yl]acetamide
methyl 3-({[3-(2-fluorophenyl)phenyl]formamido}methyl)-5-(pyridine-4-amido)benzoate
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
[(5-ethylpyridin-2-yl)methyl](methyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
ethyl 4-[3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-amido]piperidine-1-carboxylate
1-butyl-4-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazin-2-one
2-benzyl-4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1,3-thiazole
4-(azocan-1-yl)-N-(3-methoxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-hydroxy-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
1-(2-butoxybenzoyl)-2-(pyrrolidine-1-carbonyl)piperazine
1-[(3-methoxyphenyl)methyl]-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazin-2-one
2-[1-(propan-2-yl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
N-[2-(5-methylthiophen-2-yl)ethyl]-2-(3-oxopiperazin-1-yl)acetamide
5-cyclopropyl-3-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2-oxazole
3-(1,4-oxazepane-4-sulfonyl)-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
(1S,9S)-11-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
3-benzyl-4-(oxane-4-carbonyl)piperazin-2-one
N-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carboxamide
6-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carbonyl]pyridin-2-amine
5-({[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
8-[3-(2-oxoazepan-1-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
1-benzyl-N,N-dimethyl-5-(5-propyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine