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(3S)-1-[5-(4-methoxyphenyl)furan-2-carbonyl]-N,N-dimethylazepan-3-amine
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-3-(1H-1,3-benzodiazol-2-yl)propan-1-one
2-ethyl-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrimidine
N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
ethyl 5-[(4-carbamoylpiperidin-1-yl)methyl]-1-(2,4-dimethylphenyl)-1H-pyrazole-4-carboxylate
(3S,7S)-5-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]urea
3-chloro-5-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1,2-dihydropyridin-2-one
N-(furan-2-ylmethyl)-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
4-[2-(2-oxoimidazolidin-1-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(2S,4S)-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2-(propan-2-yl)pyrimidine
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
3-[(tert-butylamino)methyl]-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
9-[2-(pyridin-2-yl)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
2-(5-chloro-2-methoxypyridin-4-yl)-5-fluoro-N,N-dimethylpyrimidin-4-amine
(3S,4S)-1-[(3-methylthiophen-2-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-({5-[(3-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
5-[(3S)-3-ethylmorpholine-4-carbonyl]-2-(trifluoromethyl)-1H-1,3-benzodiazole
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
3-[(3,5-dimethylphenyl)methyl]-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(2S,4R)-1-[(2-methoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1-methylpiperidine-2-carboxamide
1-[5-(2,4-dimethylbenzoyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-(1H-1,3-benzodiazol-2-ylmethyl)-3-(3-hydroxy-3-methylbutyl)benzamide
methyl 9-[(4-fluorophenyl)methoxy]-7-oxo-3-(quinolin-8-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(3-chloro-5-fluoro-4-methoxyphenyl)-5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
7-[(3,4-difluorophenyl)methyl]-2-(pyridine-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-({[(2-chloropyridin-3-yl)methyl](methyl)amino}methyl)-6-methoxy-1,2-dihydroquinolin-2-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]acetamide
(3R,4S)-1-[2,4-bis(trifluoromethyl)benzoyl]-4-cyclopropylpyrrolidin-3-amine
3-{2-[4-(2,5-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-chloro-2-methylphenyl)urea
2-(6-methoxynaphthalen-2-yl)-4-(5-propyl-1,3,4-oxadiazole-2-carbonyl)morpholine
2-(4-acetyl-4-phenylpiperidine-1-carbonyl)pyrrolidine-1-carboxamide
1-{1-[5-(2-chlorophenyl)furan-2-carbonyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)benzamide
1-[(1-phenylcyclopropyl)methyl]piperidin-3-ol
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-2-(1-methylpyrrolidin-2-yl)acetamide
2-{1-[4-(1H-pyrazol-3-yl)benzoyl]-1,4-diazepan-6-yl}acetic acid
{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
N-[(2S)-oxolan-2-ylmethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(3-chloro-4-hydroxyphenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
2-({[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyrimidine
(2S,4S)-4-amino-1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}pyrrolidine-2-carboxylic acid
1-[6-(4-methoxypiperidin-1-yl)pyridine-3-carbonyl]-4-phenylazepane