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4-[6-(cyclopropylamino)pyridazin-3-yl]benzamide
5-(2-chlorophenyl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]furan-2-carboxamide
2-acetyl-8-(thiophen-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[2-(dimethylamino)ethyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
5-methyl-2-phenyl-N-(1-phenylethyl)-1H-imidazole-4-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl]({[2-fluoro-4-(trifluoromethyl)phenyl]methyl})methylamine
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(oxolan-2-ylmethyl)-N-propylpiperidine-4-carboxamide
6-[3-(trifluoromethyl)phenyl]-2H-1,3-benzodioxole-5-carboxamide
N-ethyl-6-(3-methoxyphenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-{4-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]piperidin-1-yl}-6-fluoro-4-methylquinazoline
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]pyridine-2-carboxamide
N-(2-methoxyethyl)-1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-(3-fluorophenoxymethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1H-pyrazole-3-carboxamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-(3-methylpyridin-2-yl)piperazine
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[1-(thiophen-2-yl)propan-2-yl]propanamide
1-methyl-4-({4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)piperazine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-ethyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
3-[3-(4-fluorophenyl)oxolan-3-yl]-5-(1H-pyrrol-2-yl)-1,2,4-oxadiazole
methyl 5-(benzylamino)-3-(furan-2-amido)-1-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-1-(oxan-4-yl)urea
ethyl 4-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
(2S,4S)-4-amino-1-(2,5-dimethoxybenzenesulfonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)propanamide
4-(2-fluoro-4-methylbenzoyl)-1-(3-methoxyphenyl)-5-methylpiperazin-2-one
3-[1-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(1-{[1-(3,6-dimethylpyrazin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-1-(pyridin-2-yl)piperidine-3-carboxamide
2-[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]benzoic acid
7-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-{4-[2-(2H-indazol-2-yl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2,6-dimethoxybenzamide
1-[4-({[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)phenyl]ethan-1-one
(2S,4R)-1-benzyl-N-[2-(dimethylamino)ethyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carboxamide
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3,3,3-trifluoropropan-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(dimethylamino)propyl]acetamide
N-methyl-N-(2-phenylethyl)-5-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}methyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-methyl-3-(2-methylpropyl)-N-[(3-methylpyridin-4-yl)methyl]-1,2-oxazole-5-carboxamide
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
3-[3-(heptan-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4-methyl-1,2,5-oxadiazole
5-methyl-3-[1-(pyridin-4-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
2-(2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-[3-(2-methoxyethoxy)phenyl]-3-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]urea
N-ethyl-7-[(oxolan-2-ylmethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethyl-1,3-oxazole-5-carboxamide
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]piperidin-4-ol
2-[1-(4-methylpyridin-2-yl)-1H-pyrazol-3-yl]pyrazine
2-(1H-1,3-benzodiazol-1-yl)-1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]ethan-1-one
2-phenyl-N-{1-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
5-methyl-4-[(oxolan-2-ylmethyl)amino]-N-(thiophen-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide