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7-fluoro-N,N-dimethyl-2-[2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-5-yl]quinoline-4-carboxamide
3-[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
4-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
N-[(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-3-fluorobenzamide
1-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
2-(3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}phenoxy)acetamide
1-(azocan-1-yl)-3-[5-methoxy-2-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
7-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1-oxa-7-azaspiro[3.5]nonane
ethyl 1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-[cyclopropyl(3-phenylprop-2-yn-1-yl)amino]-N-(1,3-thiazol-2-yl)propanamide
2-(2-methoxy-5-methylphenyl)-2-{methyl[2-(1H-pyrazol-1-yl)ethyl]amino}acetic acid
1-[2-({[(2-chlorophenyl)methyl](methyl)amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
ethyl 4-benzyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
4-(4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperazin-1-yl)-6-methylpyrimidin-2-amine
(1S,5R)-3-(3,5-dimethyl-1-benzofuran-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,4S)-4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)oxolan-3-ol
2-{4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}pyridine-4-carbonitrile
3-fluoro-N-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1-methylcyclopropyl)propan-1-one
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-2-(3-fluoro-4-methylphenyl)acetamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}azetidin-3-yl)pyridine
1-(2-chloro-4-fluoro-5-methylphenyl)-3-[2-(2-hydroxyethoxy)ethyl]urea
2-{4-[(4-methyl-1H-imidazol-5-yl)methyl]-1,4-diazepan-1-yl}-1,3-benzothiazole
6-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(methylsulfanyl)pyrimidin-4-amine
N,4-dimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidin-2-amine
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]methylamine
1-{2-methyl-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
(3aR,6aS)-5-(4-cyanobenzoyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(butan-2-yl)-2-methyl-N-(pyridin-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
1-[(3-methoxyphenyl)methyl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-one
2-cyclopropyl-3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-6-methyl-1-[(5-methylfuran-2-yl)methyl]-1,4-dihydropyridin-4-one
methyl 5-{6-[(2-fluorophenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepan-1-yl}-5-oxopentanoate
1-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}imidazolidin-2-one
(1R,5R)-6-methyl-N-[(4-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-(2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-1H-1,2,4-triazole
N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-1,2,5-thiadiazole-3-carboxamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(2-phenylethyl)amine
8-cyclopropanecarbonyl-2-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-1-methyl-1,2-dihydroquinolin-2-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(4,6-dimethylpyrimidin-2-yl)piperidine-4-carboxylic acid
3-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-3-methylurea
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,4-dimethyl-1,3-thiazole-5-carboxamide
(4aS,8aR)-6-(2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
1-[1-(methoxymethyl)cyclopentyl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]furan-3-carboxamide
1-[(3S,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)amine