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(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(1-cycloheptylpiperidin-3-yl)-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
5-(morpholin-4-ylmethyl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1,2-oxazole-3-carboxamide
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-3-carbonyl]-2,8-dimethylquinoline
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-cyclopropaneamido-N,4-dimethylbenzamide
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclopropan-1-amine
9-[3-(methylsulfanyl)butyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6-(2,3-dimethylphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
(2S)-2-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}formamido)-3-methylbutanamide
(2S,4S)-4-amino-1-(dimethylsulfamoyl)-N-ethylpyrrolidine-2-carboxamide
4-[2-(1-phenylethyl)-1H-imidazol-1-yl]benzene-1-sulfonamide
6-(1-benzothiophen-2-ylmethyl)-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
8-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
{5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]furan-2-yl}methanol
N-benzyl-2-(4,4-dimethyl-2-oxopyrrolidin-1-yl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]acetamide
5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-methoxy-3-[3-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrazine
1-(3-methyl-1,2-oxazole-5-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
[(3-chlorophenyl)methyl](methyl){2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
methyl (1S,3S,3aR,6aS)-3-(2-chloro-6-fluoro-3-methylphenyl)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(3-methylquinoxalin-2-yl)methyl]amine
2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(3-methoxypropyl)-8-[(4-methylphenyl)methyl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-5-(2-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-ethyl-4-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}piperazine-2,3-dione
1-[(3-fluorophenyl)methyl]-4-[(4-hydroxyquinolin-2-yl)methyl]piperazin-2-one
2-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
2-{[5-(1H-indol-3-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[4-(4-{[2-(3-chlorophenyl)ethyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
5-({[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]amino}methyl)-N-methylfuran-2-carboxamide
5-(2,6-difluorophenoxymethyl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(2-methoxy-2-methylpropyl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide
N-(1,2-oxazol-3-ylmethyl)-4-(pyrrolidin-1-ylmethyl)benzamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
N,2-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-thiazole-4-carboxamide
N-[2-({5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]phenyl}formamido)ethyl]acetamide
1-(oxan-4-yl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
2-({2-[1-(ethanesulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(4-propanoylphenoxy)acetamide
3-{[benzyl(methyl)amino]methyl}-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
2-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-1-(azepan-1-yl)ethan-1-one
(3R,4R)-1-[2-(1H-imidazol-2-yl)benzoyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-[4-({[(6-chloropyridin-3-yl)methyl]carbamoyl}methyl)phenyl]butanamide
N-[1-(4-{[(2,3-difluorophenyl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]oxane-4-carboxamide
4-(4-fluorophenoxy)-1-[2-(pyridin-3-yl)acetyl]piperidine-4-carboxylic acid
(1S,5R)-3-(3-propyl-1H-pyrazole-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[(3-methoxyphenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
1-[(3-methoxyphenyl)methyl]-N-methyl-6-oxo-N-(pyrazin-2-ylmethyl)piperidine-3-carboxamide