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N-(oxolan-2-ylmethyl)-2-(2-oxopiperidin-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
4-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}-2,1,3-benzoxadiazole
N-methyl-5-oxo-1-(pyridin-2-ylmethyl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrrolidine-3-carboxamide
4-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-1-(2-phenylethyl)piperazin-2-one
2-amino-N-{1,9-dioxaspiro[5.5]undecan-4-yl}-6-(propan-2-yl)pyrimidine-4-carboxamide
2-[(4-methoxyphenyl)methyl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-(2-phenylphenyl)-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperazin-2-one
1-({1-[6-(2-methoxyphenyl)pyridazin-3-yl]piperidin-3-yl}methyl)pyrrolidin-2-one
2-[3-(3-methoxyphenoxy)propyl]benzamide
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)cyclohexanecarboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-phenyl-1,2,4-triazin-3-amine
1-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-(3-chlorophenyl)-4-(1,2-oxazole-3-carbonyl)piperazin-2-one
N-(1-{4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)acetamide
3-[2-(2-methylphenyl)ethyl]-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N-cyclopropyl-1-{1-[(dimethyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl]propanoic acid
2-fluoro-5-[({[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}carbamoyl)amino]-N-methylbenzamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(1H-pyrazol-1-yl)benzamide
3-(1,3-dihydro-2-benzofuran-5-yl)-1-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]urea
6-cyclopropyl-2-[3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N,2-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
2-({[4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)phenyl]methyl}amino)ethan-1-ol
3-({1-[4-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-yl}methyl)benzoic acid
3-[(1-acetylpiperidin-4-yl)oxy]-N,N-diethyl-4-methoxybenzamide
2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-[4-(2-methylpropanamido)phenyl]acetic acid
[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(propane-2-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(furan-3-ylmethyl)-N-methyl-2-[methyl(piperidin-4-yl)amino]acetamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](furan-2-ylmethyl)(3-methylbutan-2-yl)amine
N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-2-(propan-2-yloxy)phenyl)methanol
7-[4-(4-fluorophenyl)oxane-4-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
{3-[(3-chlorophenyl)methyl]-1-(quinoxalin-2-yl)piperidin-3-yl}methanol
6-{4-[1-(dimethylamino)ethyl]phenyl}-2-(pyrrolidin-1-yl)pyrimidin-4-amine
3-ethyl-1-({1-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-3-yl}methyl)urea
3-{[(2-hydroxy-3-methylphenyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(thiophen-3-ylmethyl)acetamide
1-cyclobutyl-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[2-(3-methoxyphenyl)acetyl]-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
[(3R,5R)-5-[(dimethylamino)methyl]-1-[4-(5-methylfuran-2-yl)benzoyl]piperidin-3-yl]methanol
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-(4-methoxyphenyl)-2-methylpiperazine
1-[3-(2-methylphenyl)phenyl]-N-[(2R)-oxolan-2-ylmethyl]piperidin-4-amine
N-[(3R,4S)-4-cyclopropyl-1-(furan-2-carbonyl)pyrrolidin-3-yl]thiophene-2-carboxamide
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
3-acetamido-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}propanamide
4-cyclopropyl-6-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
7-[(2-fluoro-5-methoxyphenyl)methyl]-6-oxo-N-propyl-2,7-diazaspiro[4.5]decane-2-carboxamide