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3-[3-(methoxymethyl)piperidin-1-yl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazine
1-methyl-3-[2-(2-methyl-4-phenylpiperazin-1-yl)-2-oxoethyl]-3-(4-phenylphenyl)pyrrolidine-2,5-dione
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-(cyclopropylmethyl)-N-propylacetamide
(3-{2-[1-(4-fluoro-3-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-(2-oxoimidazolidin-1-yl)-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)acetamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
(3S,4S)-4-cyclopropyl-1-(4-ethyl-5-methylthiophene-3-carbonyl)pyrrolidine-3-carboxylic acid
1-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N2,N2,N4,5,6-pentamethyl-N4-(pyrazin-2-ylmethyl)pyrimidine-2,4-diamine
3-[1-(1-methyl-1H-indole-4-carbonyl)piperidin-3-yl]benzoic acid
1-(6-cyclopropylpyrimidin-4-yl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
2-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)-1-(pyrrolidin-1-yl)ethan-1-one
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-(2-methyl-2H-1,2,3-triazol-4-yl)propanamide
3-(4-{[4-(difluoromethoxy)phenyl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
(1S,5R)-6-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-1-(benzenesulfonyl)-4-[4-(2-methoxyphenoxy)piperidin-1-yl]pyrrolidin-3-ol
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,5-difluorobenzamide
N-[(3R,4S)-1-(1-acetylpiperidin-4-yl)-4-cyclopropylpyrrolidin-3-yl]-2-methylfuran-3-carboxamide
N4-[3-(3,4-dimethoxyphenyl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
8-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2,5-dimethylfuran-3-carboxamide
1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-4-(pyridin-4-yl)piperazine
2-(pyridin-2-ylmethyl)-9-[6-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(3,4-difluorophenyl)-1-(1,2-oxazol-3-ylmethyl)piperidin-3-amine
N1-(prop-2-en-1-yl)-N2-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-1,2-dicarboxamide
1-(4-ethylpiperazin-1-yl)-3-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]propan-1-one
2-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-3-[4-(trifluoromethyl)benzoyl]piperidine
4-({6-chloro-4-[(2-methoxyethyl)amino]quinazolin-2-yl}methyl)-1-phenylpiperazin-2-one
4-{5-[1-(1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}thiomorpholine
N-(5-tert-butyl-1,2-oxazol-3-yl)-2-[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]acetamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
3,3-dimethyl-1-({5-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
N-{[5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
4-{1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl}benzoic acid
N-(2,4-difluorophenyl)-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-(butan-2-yl)-N3-ethyl-4-oxo-N5-[(4-phenyloxan-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-[(2-fluorophenyl)methyl]piperidin-3-amine
(4-{[methyl({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amino]methyl}oxan-4-yl)methanol
8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-cyclopentyl-3-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}-3-(3-fluorophenyl)pyrrolidine-2,5-dione
1-(2,2-difluorocyclopropanecarbonyl)-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
5-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-benzyl-1,3-thiazole-4-carboxamide
methyl 1-[(3S,5S)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[2-(dimethylamino)ethyl]-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-oxo-1-phenylpyrrolidine-3-carboxamide
2-[methyl({[2-(pyrrolidin-1-ylmethyl)phenyl]methyl})amino]acetic acid