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methyl 2-hydroxy-5-{12-oxo-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-14-yl}benzoate
2-(3-phenylpropyl)-4-(pyrazin-2-yl)morpholine
methyl 1-[(3S,5S)-1-[(2E)-3-phenylprop-2-en-1-yl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(4-ethoxyphenyl)methyl](2-methoxyethyl)amine
N,N-dimethyl-5-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-3-azaspiro[5.5]undecan-9-amine
9-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
(2S)-N-(furan-2-ylmethyl)-2-methoxy-N-[2-(morpholin-4-yl)ethyl]-2-phenylacetamide
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}({[4-(methylsulfanyl)phenyl]methyl})amine
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(4-methyl-3-phenylpiperazin-1-yl)ethan-1-one
(3S,4R)-1-[4-methoxy-3-(morpholin-4-yl)benzoyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyrazine-2-carboxamide
9-(2-cyclopropylpyrimidine-5-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
3-[2-(4H-1,2,4-triazol-4-yl)phenyl]-1,3-oxazolidin-2-one
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-4-fluoro-N-(pyridin-4-ylmethyl)benzamide
(3S,5R)-1-benzyl-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
7-(3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-[2-(methylsulfanyl)pyrimidin-4-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
N-[(1R)-1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propyl]acetamide
8-(cyclohexylmethyl)-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-ethyl-5-(4-phenyl-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazol-5-yl)-1H-1,2,4-triazole
1-(ethanesulfonyl)-4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]piperazine
4'-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(propan-2-yl)-5-(thiomorpholine-4-carbonyl)-1,3-benzoxazole
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
3-{2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2,4-difluoro-N-methylbenzamide
N-methyl-4-{1-[2-(pyrazin-2-yl)ethyl]-1H-imidazol-2-yl}benzene-1-sulfonamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
3-{[(propan-2-yl)amino]methyl}-1-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-[4-(4-{[2-(4-fluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)furan-2-carboxamide
2-(1-propylpiperidin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
5-(2-butyl-1H-imidazol-4-yl)-1-[3-(1H-imidazol-1-yl)propyl]-4-phenyl-1H-imidazole
1-(6-chloropyridazin-3-yl)-N-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-amine
(3S,4R)-1-(5-chloropyridine-3-carbonyl)-4-methylpiperidine-3,4-diol
6-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1H-indazole
2-[(1S,5R)-6-(2,3-difluoro-6-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-(2-ethyl-4-methyl-1,3-thiazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
6-{3-[2-(methylsulfanyl)ethyl]-1-propyl-1H-1,2,4-triazol-5-yl}quinoxaline
3-{1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-chlorophenyl)urea
1'-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}spiro[indene-1,4'-piperidine]
1-methyl-3-(thiophen-2-yl)-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1H-pyrazole-5-carboxamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
3-hydroxy-3-{[(propan-2-yl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-methyl-4-{5-[(2-phenylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrazole
(2S)-N-benzyl-2-(methylamino)-N-(1,3-thiazol-2-ylmethyl)propanamide