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1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrimidin-2-amine
1-cyclopentyl-6-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine-3-carboxamide
4-[5-(2-methylpropyl)-1H-1,2,4-triazol-3-yl]benzamide
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-3-phenoxypropan-1-one
1-(4-chlorophenyl)-3-cyclopropyl-5-{[1,2,4]triazolo[1,5-a]pyrimidin-6-ylmethyl}-1H-1,2,4-triazole
(1S,5R)-6-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-(3-chloro-4-methoxyphenyl)-3-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]propanamide
5-chloro-6-[3-(2-methoxyphenoxy)azetidin-1-yl]pyridine-3-carboxylic acid
2-amino-4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
1-(oxolane-2-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-methyl-2-[3-(4-methyl-3-oxopiperazine-1-carbonyl)phenyl]-1,2-dihydrophthalazin-1-one
1-({4-[(5-methylpyridin-3-yl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
methyl 4-({4-[2,5-dioxo-4-(2-phenylethyl)imidazolidin-4-yl]piperidin-1-yl}methyl)benzoate
(3aR,5S,6S,7aS)-2-[(4-hydroxy-6-methylquinolin-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
2-{4-[1-(carbamoylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-cyclohexylacetamide
(3S,4R)-3-benzyl-4-methyl-1-(3-methylpyrazin-2-yl)piperidin-4-ol
4-{2-[(5-chloropyrimidin-2-yl)oxy]hex-5-en-1-yl}morpholine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}({[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl})methylamine
6-fluoro-2-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}quinolin-4-ol
2-methoxy-5-{1-[1-(thiophen-3-yl)propan-2-yl]-1H-imidazol-2-yl}pyrimidine
4,6-dimethyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyridine-3-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(pyridin-4-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
ethyl 4-(4-{4-[(1,4-dioxan-2-ylmethyl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
3-(3-methoxypropyl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
N-cycloheptyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
3-{5-[2-(pyrrolidin-3-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
2-{[({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)amino]methyl}-6-methyl-3,4-dihydropyrimidin-4-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(propan-2-yl)acetamide
(4aS,7aR)-1-[(3-chloro-4-hydroxyphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
5-(furan-3-yl)-1-(1-phenylethyl)-1H,4H-pyrazolo[3,4-d]imidazole
1-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-(1H-indol-1-ylmethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-(dicyclopropylmethyl)-N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-cyclohexyl-N-(2-methanesulfonamidoethyl)-1H-pyrazole-4-carboxamide
(1R,5S,8R)-3-[(3-chloro-4,5-diethoxyphenyl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
3-(2-cyanophenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-methyl-N-[2-(oxan-4-yl)ethyl]-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetamide
4,6-dimethyl-1-(2-{[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
3-(methylsulfanyl)-1-{4-[3-oxo-3-(4-phenylpiperazin-1-yl)propyl]piperidin-1-yl}propan-1-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(3-methylphenyl)methyl](oxolan-2-ylmethyl)amine
3-[5-(2,4-difluoro-3-methoxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
4-{2-[1-(pyridine-3-sulfonyl)piperidin-2-yl]ethyl}morpholine
1-[(2-methoxyphenyl)methyl]-6-oxo-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}piperidine-3-carboxamide
1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(3-methoxypropyl)piperidine
7-(1-benzothiophen-3-yl)-9-ethoxy-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[4-({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)-1,4-diazepan-1-yl]ethan-1-one