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methyl (2S,4S)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-[4-(3-fluorophenyl)benzamido]pyrrolidine-2-carboxylate
5-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-(2-methoxyethyl)-1,2,4-oxadiazole
N-cyclopropyl-1-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}piperazine-2-carboxamide
4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole
2,2-dimethyl-N-[(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)methyl]propanamide
2-[2-(dimethylamino)ethyl]-9-{[2-(ethylamino)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
3-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}azetidin-3-yl)pyridine
4-ethyl-1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1,4-diazepan-5-one
N,5-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
1-[2-({[2-(dimethylamino)-6-ethylpyrimidin-4-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
5-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-2,1,3-benzothiadiazole
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(oxan-2-ylmethoxy)acetamide
4-[4-(3-chloro-4-fluorophenyl)piperazine-1-carbonyl]-1-[2-(dimethylamino)ethyl]pyrrolidin-2-one
2-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}-2-oxoethyl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-N-(1,3-thiazol-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)benzamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-(1-phenylpiperidin-4-yl)acetamide
(1,3-benzothiazol-2-ylmethyl)({[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
2-chloro-N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-5-acetamidobenzamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine
4-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-(dimethylamino)-N-methyl-2-(2-methylphenyl)acetamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-[(1-ethylpiperidin-4-yl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
2-(5-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}thiophen-2-yl)-1H-imidazole
7-(2,2-dimethylpropyl)-2-[(trimethylpyrazin-2-yl)methyl]-2,7-diazaspiro[4.5]decane
1-{[2-(2-aminopyrimidin-5-yl)phenyl]methyl}piperidin-4-one
1-(2,3-dihydro-1H-inden-2-yl)-4-(5-ethyl-1,3,4-oxadiazol-2-yl)piperazine
1-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
[1-(piperidin-3-yl)piperidin-4-yl]methanol
(3S,7S)-5-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-triene-3-carboxylic acid
N-{2-[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclobutanecarboxamide
N-[(3-fluorophenyl)methyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}piperidin-2-one
5-propyl-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-[1-butyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-2,2-dimethylthiomorpholin-3-one
2-[(5-hydroxy-6-methyl-1,2,4-triazin-3-yl)sulfanyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
2-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-phenylcyclopent-2-en-1-one
2-(3-methylphenyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(1S,4R)-1-({[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]sulfonyl}methyl)-7,7-dimethylbicyclo[2.2.1]heptan-2-one
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-2-carboxamide
1-(1,4-dioxan-2-ylmethyl)-1-methyl-3-(2,4,6-trimethylpyridin-3-yl)urea
1-{[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
4-[(1-methyl-1H-imidazol-5-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
9-(5-methyl-1,3-oxazole-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1'-[(2-aminopyridin-3-yl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one