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N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
7-(2-hydroxyethyl)-2-[3-(pyridin-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-methyl-4-(2-methyl-1,6-naphthyridine-3-carbonyl)piperazin-2-one
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-one
3-(azocan-1-yl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]propanamide
2-{2-[2-(2-methoxyphenyl)-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
ethyl 3-[(2-fluorophenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-3-carboxylate
5-(4-benzylpiperidine-1-carbonyl)-1-(butan-2-yl)-N-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(2-hydroxyethyl)-9-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[3-(pyrrolidin-1-yl)pyrazin-2-yl]-1H-indole
(1R,9S)-5-amino-3-[4-(1H-imidazol-1-yl)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
N-({1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
1'-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
N-[5-carbamoyl-2-(3-methylpiperidin-1-yl)phenyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
4-[1-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-imidazol-2-yl]-5-methyl-2-(thiophen-2-yl)-1,3-oxazole
1-(2-phenylethyl)-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,9aR)-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(cyclohexylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
N-[2-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)ethyl]acetamide
1-[(2,3-difluorophenyl)methyl]-4-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]piperidine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(pyridin-3-yl)propan-1-one
ethyl 2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
3-[5-(2,1,3-benzoxadiazol-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-(4-ethyl-3,3-dimethylpiperazin-1-yl)-N-(2-fluoro-5-methylphenyl)-4-oxobutanamide
1-[(4-fluorophenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-{4-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-1,2,3-triazol-1-yl}propanoic acid
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[(2-methylpropyl)amino]methyl}piperidin-2-one
3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}urea
methyl 6-oxo-4-[2-(propan-2-yl)-1,3-oxazol-4-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2R,3R)-3-(morpholin-4-yl)-1'-(oxan-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3,5-dimethyl-N-(3-methyl-1-{7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)benzamide
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetic acid
N-(1,1-dioxo-1λ6-thiolan-3-yl)-2,6-dimethyl-N-(prop-2-en-1-yl)quinoline-4-carboxamide
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
N-[2-(2,5-dimethylphenyl)ethyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
3,3,3-trifluoro-1-{3-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}propan-1-one
(1R,9aR)-1-[(4-benzoylpiperidin-1-yl)methyl]-octahydro-1H-quinolizin-1-ol
ethyl 5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-imidazole-4-carboxylate
N-(5-acetamido-2-fluorophenyl)-2-[(methylcarbamoyl)methyl]-3-oxopiperazine-1-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-(morpholin-4-ylmethyl)piperidin-2-one
3-(3,4-difluorophenyl)-5-(5-methoxyfuran-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-{3-[1-(3,3,3-trifluoro-2-hydroxypropyl)-1H-imidazol-2-yl]phenoxy}acetamide
4-chloro-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
(3S,4R)-1-(1-acetylpiperidine-4-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)-2-methanesulfonylacetamide
3-cyclopropyl-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
4-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine