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7-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
2-{1-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-N-ethylformamido}propanamide
dimethyl({3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]propyl})amine
2-[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]acetamide
1-(4-ethylpiperazin-1-yl)-3-[3-({[3-(pyridin-3-yloxy)propyl]amino}methyl)phenoxy]propan-2-ol
4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
1-(4-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-3,5-dimethyl-1H-pyrrol-2-yl)ethan-1-one
(3S,4R)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
5-cyclobutyl-N-[1-(cyclohex-1-en-1-yl)ethyl]-1,3,4-oxadiazol-2-amine
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-4-(pyrrolidine-1-carbonyl)pyridine
2-amino-4-[2-(2-hydroxyethoxy)phenyl]-6-(4-methylphenyl)pyridine-3-carbonitrile
3-{[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]amino}-1-(morpholin-4-yl)propan-1-one
2-methoxy-4-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
1-[2-(2-phenylethyl)morpholin-4-yl]-3-(1H-pyrazol-4-yl)propan-1-one
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methylbutanamide
11-(cyclooctylamino)-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
N-cyclopropyl-3-fluoro-N-({4-methoxy-3-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)benzamide
N-{1-[1-(4-fluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
4-[3-(2,2-dimethylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-propyl-1,3-thiazole
propan-2-yl 2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxylate
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
5-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
N-methyl-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
2-[5-(3-methoxypyrazin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
4-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
N-[3-(azepan-1-yl)-2-hydroxypropyl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
3-(2-fluorophenyl)-5-(thiophen-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
1-methyl-N-{3-[(5-methylpyridin-2-yl)amino]propyl}azepane-2-carboxamide
2-ethyl-5-{[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}pyrimidine
4-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
4-{4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-benzyl-5-[4-(2-methoxyphenyl)piperazin-1-yl]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-cyclopropyl-2,2-dimethyl-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)oxane-4-carboxamide
{5-fluoro-7-[5-(2-methylpropyl)-1H-1,2,4-triazol-3-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-[({[1-(2-methoxyethyl)piperidin-3-yl]methyl}(methyl)carbamoyl)amino]benzamide
4-(4-methylpiperazin-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pentan-1-one
1-(5-methoxy-2-{[(2-phenoxyethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
2-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-5-methoxy-4H-pyran-4-one
1-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-1-methyl-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)urea
4-methyl-3-{10-oxo-3,9-diazaspiro[5.6]dodecane-3-carbonyl}benzene-1-sulfonamide
1-(3-{[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]methyl}phenyl)ethan-1-one
3-[4-(3-cyanopyridin-2-yl)piperazin-1-yl]-N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)propanamide
(2R,3R,6R)-5-(cyclopropanesulfonyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3-hydroxyphenyl)ethan-1-one
[4-methyl-5-(1-{[2-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methanol
3-{2-[5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methyl-4H-1,2,4-triazole
(4-{[(5-methylpyrazin-2-yl)methyl]amino}quinazolin-2-yl)methanol