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1-benzyl-3-(pyridin-2-ylmethyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrimidin-2-amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-methylpiperidine
5-{2-azaspiro[4.4]nonane-2-carbonyl}-N-ethylpyrimidin-2-amine
1-[1-(4-cyanopyridin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
(1R,3S,5S)-8-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane
7-chloro-3-[1-(pyridin-3-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-(3-carbamoylpyridin-2-yl)-4-(3-phenylpropyl)piperidine-4-carboxylic acid
3-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-1-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
1-[(3-methoxyphenyl)methyl]-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
9-(2-fluoro-2-phenylacetyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methyl-6-propylpyrimidine
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-4-(piperidin-1-yl)butanamide
(2R)-2-amino-1-[2-amino-4-(1,4-oxazepan-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]propan-1-one
3-(dimethyl-1,3-thiazol-5-yl)-2-methoxypyridine
N1-(3-methylpyridin-4-yl)-N2-[6-(propan-2-yl)pyrimidin-4-yl]ethane-1,2-diamine
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
3-(2-methyl-1H-imidazol-1-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]propanamide
N,N-dimethyl-2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetamide
2-[4-(6-phenylpyridazin-3-yl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
5-{1-[(2E)-2-methylbut-2-enoyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
4-[3-cyclopropyl-5-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethyl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
1-(oxolane-2-carbonyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-amine
ethyl 1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(3-fluorophenyl)methyl]piperidine-4-carboxylate
1-(1H-imidazol-2-ylmethyl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
5-{4-[(2-phenylazetidin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
N-[(3S,4R)-1-(1,3-benzoxazol-2-yl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
3-{3-[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]propyl}-1H-indole
1-(1H-imidazol-2-ylmethyl)-3-(2-methylphenyl)pyrrolidin-3-ol
3-{1',5',6',7'-tetrahydrospiro[cyclohexane-1,4'-imidazo[4,5-c]pyridine]-5'-ylmethyl}-4H-chromen-4-one
1-(4-fluoropiperidin-1-yl)-2-{4-[(4-phenylphenyl)methyl]morpholin-3-yl}ethan-1-one
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(2-phenylethyl)piperazine
2-(3-hydroxypropyl)-9-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine
methyl 3-{[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}propanoate
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-methyl-1,3-benzothiazole-6-sulfonamide
N-[(3S,7S,8aS)-3-(cyclohexylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
2-{4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-2-fluoro-5-methylbenzene-1-sulfonamide
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
4-(4-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
5-methoxy-3-methyl-2-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}-1H-indole
methyl[2-(1H-pyrazol-4-yl)ethyl][(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
(3aR,6aR)-2-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-indazol-3-yl)acetamide
5-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrazine-2-carboxamide
4-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-methyl-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-cyclohexyl-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one