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N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
(2S,4R)-1-[(2,5-dimethylphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
2-[N-(4-methylphenyl)methanesulfonamido]-N-(2-phenoxyethyl)acetamide
2-methoxy-5-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-ylmethyl]benzoic acid
2-[2-(4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperazin-1-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
(3R,4R)-4-(azepan-1-yl)-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-ol
2-amino-6-{3-[1-(dimethylamino)ethyl]phenyl}pyrimidin-4-ol
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(1,2-oxazol-3-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
8-[(3E)-pent-3-enoyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
7-(5-chloropyridin-2-yl)-4-(pyrimidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[6-(methoxymethyl)pyrimidin-4-yl]pyrrolidin-3-yl]methanol
2-(3-chloro-4-hydroxyphenyl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}acetamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(4-methyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(4-fluoro-2-methoxyphenyl)methyl]-2-[(3-methoxyphenyl)methyl]morpholine
N-(butan-2-yl)-N-cyclopentyl-2-(4-methanesulfonylphenyl)acetamide
3-{[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}quinolin-7-ol
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)amino]propane-1,3-diol
(3S,4S)-1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
4-(5-{[(2-chlorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)-N-(prop-2-en-1-yl)piperidine-1-carboxamide
4-{3-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]phenyl}morpholine
1-[(4-chlorophenyl)methyl]-4-(3,5-difluoropyridine-2-carbonyl)piperazine
N-cyclobutyl-4-{2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]acetyl}morpholine-2-carboxamide
1-(3-chlorophenyl)-4-{4-[(2-hydroxyethyl)(methyl)amino]benzoyl}piperazin-2-one
[(3R,4R)-1-(4-chloro-1H-indole-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]-2-methyl-1,4-diazepan-5-one
{[3-(azocane-1-carbonyl)-1,2-oxazol-5-yl]methyl}(benzyl)methylamine
N-[2-(4-methoxyphenyl)ethyl]-2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carboxamide
4-ethyl-3-{[1-(2-methyl-2-phenoxypropanoyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-{[4-(3-chlorophenyl)-5-{[methyl({[4-(trifluoromethoxy)phenyl]methyl})amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
(2R,6R)-4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(2-fluorophenyl)-4-[(2,3,4-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)-4-(4-methoxyphenyl)piperazine
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
1-cyclopentyl-5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
1-benzyl-N3-[2-(4-chlorophenyl)ethyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[1-(1-{[3-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-2-phenylethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
2-cyclopropyl-9-(2-methoxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-cyclopropyl-N-(2,3-dihydro-1H-inden-2-yl)-5-oxo-N-propylpyrrolidine-3-carboxamide
N-{4-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}acetamide
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(3-fluorophenyl)methyl]benzamide
4-benzyl-3-ethyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-1,4-diazepan-5-one
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(4-fluorophenyl)ethan-1-one
1-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}azocane
(2S)-3-hydroxy-2-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}propanamide
1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]cyclopropane-1-carboxamide