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N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(furan-2-ylmethyl)benzamide
2-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amino}methyl)-6-methylpyridin-3-ol
(3aR,6aR)-2-cyclobutanecarbonyl-5-(5-methyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-methylbut-2-enamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(1,4-dioxan-2-ylmethyl)-N-methyl-2-(1-methyl-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-4-yl)acetamide
2-{2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
3-benzyl-8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[3-(4-fluorophenyl)propyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(4-ethylpiperazin-1-yl)-3-[3-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-ethyl-5-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
6-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
N-(2-{7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
2-(3-chlorophenoxy)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)acetamide
(1S,4S)-5-[1-(4-chlorophenyl)cyclobutanecarbonyl]-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-ethyl-5-(1-ethyl-1H-pyrazol-3-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
1-({1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-[2-(4-fluorophenyl)ethyl]-N-({2-[3-(hydroxymethyl)piperidin-1-yl]-7-methoxyquinolin-3-yl}methyl)propanamide
1-phenyl-N-{[1-(quinolin-8-ylmethyl)piperidin-3-yl]methyl}methanesulfonamide
5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-N-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(oxan-4-ylmethyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(2,2-dimethylpropyl)piperidine-4-carboxamide
2-(thiophen-2-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1,3-thiazole-4-carboxamide
4-({4-[4-(2-fluorophenyl)piperazine-1-carbonyl]furan-2-yl}methyl)morpholine
N-benzyl-3-[1-(furan-2-carbonyl)piperidin-4-yl]-N-methylpropanamide
7-fluoro-N,2-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]quinoline-4-carboxamide
(4-methoxy-4-methylpentan-2-yl)[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amine
4-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1-oxaspiro[4.4]nonan-2-one
9-(2-methyloxolane-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{4-[1-(3,4-dimethoxyphenyl)-1H-imidazol-2-yl]phenyl}acetamide
2-[(2-chlorophenyl)methyl]-4-{4-[1-(2-phenylethyl)piperidin-4-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
(4aS,7aR)-1-(3-chloro-4-methylbenzoyl)-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-chloro-2-methyl-N-[(3R)-piperidin-3-yl]quinoline-4-carboxamide
2-[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-3-(piperidine-1-carbonyl)pyrazine
(3R,4R)-3-[ethyl({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]-4-hydroxy-1λ6-thiolane-1,1-dione
1-(5-ethoxyfuran-2-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
3-cyclobutyl-4-[2-(methylsulfanyl)ethyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1R,2S)-2-[1-(2,4-difluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-N-propylcyclohexane-1-carboxamide
5-(2-chloro-4-fluorophenoxymethyl)-N-[2-(propan-2-yloxy)ethyl]-1,2-oxazole-3-carboxamide
N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-{2-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]pyrimidin-4-yl}piperidin-4-ol
4-{1-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-imidazol-2-yl}pyridine
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(4-methylphenoxy)ethyl]amine
8-(dimethyl-1,3-oxazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-2-azaspiro[4.4]nonane
2-[(1-cyclopropanecarbonylpiperidin-4-yl)formamido]-3-(1H-imidazol-4-yl)propanoic acid
methyl 1-{[4-(4-acetyl-1,4-diazepan-1-yl)-8-methylquinazolin-2-yl]methyl}piperidine-2-carboxylate
2-(3,4-dichlorophenyl)-4-[(4-methoxypyridin-2-yl)methyl]morpholine