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4-{3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}pyridine
4,6-dimethyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidine
5-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
N-[(3S,4R)-1-[(2,4-difluorophenyl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
2-{[({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]methyl}-5-methoxyphenol
[3-benzyl-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-3-yl]methanol
(3aR,7aS)-5-methyl-2-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)quinoxaline-6-carboxamide
(4aR,8aS)-6-[(4-ethoxyphenyl)methyl]-1-[2-(2-fluorophenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[(2,4-difluorophenyl)methyl]-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]propanamide
1-(cyclohexylmethyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(3S,4S)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
2,6-dimethyl-4-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)phenyl acetate
1-[1-(3-fluoropyridin-4-yl)piperidin-4-yl]-2-phenylethan-1-ol
1-(4-phenylphenyl)-N-(piperidin-4-yl)piperidin-4-amine
1-(cyclohexylmethyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]piperidin-2-one
1-(pyrimidin-2-ylmethyl)-1,2,3,4-tetrahydroquinolin-2-one
2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinolin-5-ylmethyl)acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[1-(piperidin-1-yl)cyclohexyl]methyl}amine
N-{[2-(diethylamino)pyridin-3-yl]methyl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
3-(1H-imidazol-1-yl)-4-methylbenzamide
2-[2-(1,4-oxazepan-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]quinoxaline
6-(benzyloxy)-1-cyclohexyl-4-(pyrazine-2-carbonyl)-1,4-diazepan-2-one
2-(4-fluorophenyl)-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
2-ethyl-8-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
6-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-N,N-dimethylpyrazine-2-carboxamide
N-[3-(4-chlorophenoxy)propyl]-3-(3-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-propylacetamide
(4aS,7aR)-4-benzyl-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-1-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}ethan-1-one
2-(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
methyl 9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-3-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N4-methyl-N2-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-5H,6H,7H-cyclopenta[d]pyrimidine-2,4-diamine
N-cyclopropyl-5-(quinoxalin-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
4-[2-(4-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]morpholine
5-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-methyl-2-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
1-[2-(3-methoxyphenyl)ethyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
N-(5-chloro-2-methoxyphenyl)-3-[(4-methylpiperazin-1-yl)methyl]piperidine-1-carboxamide
3-[5-acetyl-2-(morpholin-4-yl)phenyl]propanamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2,6-dimethylpyridine-4-carbonyl)pyrrolidin-3-yl]methanol
2-(4-acetylpiperazin-1-yl)-N-(1H-1,3-benzodiazol-2-yl)acetamide
{1-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperidin-3-yl}methanol
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-(2-methylprop-2-en-1-yl)pyridin-2-amine
4-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1,4-oxazepan-5-one
2-{4-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine