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2-cyclopentyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2-phenyl-N-(pyridin-2-ylmethyl)acetamide
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]urea
8-[(3,4-dimethoxypyridin-2-yl)methyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)butane-1-sulfonamide
N-[(2R,3R)-2-methoxy-1'-[3-(1H-pyrazol-1-yl)propyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
3,5-dimethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]furan-2-carboxamide
3-methoxy-N-[1-(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]propanamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
N-(cyclopropylmethyl)-5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
(1S,5R)-6-(3-methylbenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 3-(2-chlorobenzenesulfonamido)-5-[(2-cyclopentylacetamido)methyl]benzoate
methyl 5-{[(4-ethoxyphenyl)methyl]amino}-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(2,6-dimethylpyridin-4-yl)-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
N-(2-phenylethyl)-4-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]oxy}benzamide
(2E)-N-[(7-{imidazo[1,2-a]pyridine-2-carbonyl}-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(thiophen-2-yl)prop-2-enamide
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
5-(methoxymethyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}furan-2-carboxamide
1-{4-[2-(2,4-dimethoxy-3-methylphenyl)-1H-imidazol-1-yl]phenyl}-1H-1,2,3,4-tetrazole
N-(1,3-dihydro-2-benzofuran-5-yl)-5-(1-propanoylpyrrolidin-2-yl)thiophene-2-carboxamide
4-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}-2-(trifluoromethyl)morpholine
N,N-dimethyl-1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-amine
2-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}pyridine-3-carbonitrile
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
4-methyl-3-oxo-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-3,4-dihydroquinoxaline-2-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
N-{[1-(2,4-dimethoxybenzenesulfonyl)piperidin-3-yl]methyl}furan-2-carboxamide
2-(5-{1-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazol-3-yl)pyridine
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-(2-methylpropyl)piperidin-4-amine
2-({[(3R,4S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]carbamoyl}methoxy)acetamide
7-(2-hydroxyethyl)-2-(4-oxo-4H-chromene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(furan-2-yl)propan-1-one
3-[(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-6-methyl-4H-chromen-4-one
3-{2-[4-(2-hydroxyphenyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
5-ethyl-5-{1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[3-(trifluoromethyl)phenoxy]piperidine
N,N-diethyl-2-(4-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)acetamide
ethyl 5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1H-pyrazole-4-carboxylate
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
1-(3-methoxypropyl)-8-(4-methylpentan-2-yl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-indol-3-yl)ethyl]acetamide
N,1-dimethyl-N-[2-(morpholin-4-yl)propyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-8-methyl-2,8-diazaspiro[5.5]undecane
2-{[4-(3-chlorophenyl)-5-(piperidin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-5-methylthiophene-2-carboxamide
1-acetyl-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-[5-(5-fluoro-3,8-dimethylquinolin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N'-cyclopentyl-N-[2-(methylsulfamoyl)ethyl]butanediamide