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(3S,9aR)-8-(2,5-difluorobenzoyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4S)-4-cyclopropyl-1-(3-fluoro-4-methylbenzoyl)pyrrolidine-3-carboxylic acid
N-[2-(diethylamino)ethyl]-N-ethyl-3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carboxamide
4-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-1-ethyl-1,2-dihydropyridin-2-one
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[(1R,2S)-2-phenylcyclohexyl]propanamide
1-(2-cyclohexylethyl)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(pyrrolidine-1-sulfonyl)piperazine
5-(3-ethylpiperazine-1-carbonyl)-2,3-dimethyl-1H-indole
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[2-(3-methoxyphenyl)ethyl]amine
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-(ethanesulfonyl)ethyl]benzamide
2-[4-(3-chlorophenyl)-2-methyl-5-oxopiperazin-1-yl]-N-(furan-2-ylmethyl)acetamide
2-(2,5-dioxoimidazolidin-4-yl)-N-[(4-phenyloxan-4-yl)methyl]acetamide
5-[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]pyridin-2-amine
3-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-2,4-dichlorophenol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,2,3-trimethylquinoxaline-6-carboxamide
3-methyl-6-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]pyridazine
N-(4-tert-butyl-1,3-thiazol-2-yl)-2-{[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]amino}acetamide
{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-(2-phenylethyl)piperidin-4-yl}methanol
1-{3-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
4-chloro-1-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
2-{3-[2-(pyridin-3-yl)-1H-imidazol-1-yl]propyl}-1,3-benzothiazole
1-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-1,2,3,6-tetrahydropyridazine-3,6-dione
N-(3,4-dimethoxyphenyl)-3-[(3S,4R)-4-(dimethylamino)-1-(2,2-diphenylethyl)piperidin-3-yl]propanamide
1-(4-chloro-2-ethylphenyl)-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3,4,5-trimethoxybenzamide
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-3-carboxamide
8-[2-(3,5-difluorophenyl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
dimethyl[2-({1-[1-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}oxy)ethyl]amine
3-(2H-1,3-benzodioxol-5-yl)-1-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1-methylurea
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]-3-hydroxypyridine-2-carboxamide
(4aR,7aS)-1-(2-methylpropyl)-4-(1,2-oxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-N-(cyclohexylmethyl)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carboxamide
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]-5-methylphenol
1-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
N-methyl-5-oxo-1-[4-(propan-2-yl)phenyl]-N-[(5-propyl-1H-pyrazol-3-yl)methyl]pyrrolidine-3-carboxamide
2-amino-N-[(3R,4S)-4-cyclopropyl-1-(dimethylcarbamoyl)pyrrolidin-3-yl]-6-(2-methylpropyl)pyrimidine-4-carboxamide
2-[(1S,5R)-3-(1H-imidazole-2-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-(2,5-dichlorophenyl)-6-methoxypyrimidin-2-amine
4-oxo-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
(2S,4S)-4-cyclopentaneamido-N,N-diethyl-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidine-2-carboxamide
11-{[(2,5-difluorophenyl)methyl]amino}-4-(3-methoxypropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1-methyl-N-(2-methylpropyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1H-indol-3-yl)acetamide
6-methyl-N-(oxolan-3-ylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)cyclohexanecarboxamide
N1-(4-methylpyridin-2-yl)-N2-[1-(oxolane-2-carbonyl)piperidin-4-yl]ethane-1,2-diamine
3-benzyl-8-[(5-methylthiophen-2-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one