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(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-ol
N-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}-1-(trifluoromethyl)cyclopropane-1-carboxamide
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-phenoxyethan-1-one
methyl 2-[1-(1,3-benzothiazole-2-carbonyl)-3-oxopiperazin-2-yl]acetate
(4aR,7aS)-1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(4-fluorophenyl)methyl]-5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-4,5-dihydro-1,2-oxazole
(3R,4S)-4-(4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)oxolan-3-ol
1,9-dimethyl-4-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(2-hydroxyethyl)-5-[3-(5-methylfuran-2-yl)butyl]-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-3-(1-methyl-1H-pyrazol-4-yl)urea
N-[(3R)-piperidin-3-yl]-2-(4H-1,2,4-triazol-4-yl)benzamide
{3-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]phenyl}methanol
2-amino-6-{4-[2-(benzyloxy)ethyl]piperazin-1-yl}pyrimidin-4-ol
3-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propanamide
3-({4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}methyl)phenol
(3R,4R)-1-(furan-3-ylmethyl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
4-chloro-N-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
N-[2-(2-fluorophenyl)ethyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
(butan-2-yl)(3-methylbut-2-en-1-yl)(pyridin-4-ylmethyl)amine
4-(1-ethyl-1H-pyrazole-3-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
1-(4-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one
N-(1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
5-(3-methoxyphenyl)-4-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-2-(pyridin-4-yl)pyrimidine
4-oxo-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-4H-chromene-3-carboxamide
3-({4-[4-(piperidin-3-yl)benzoyl]piperazin-1-yl}methyl)phenol
2-{2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-4-carbonitrile
1-(2-methoxyphenyl)-4-[4-(morpholin-4-yl)pentanoyl]piperazin-2-one
3-(2-{[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-(2-chloro-6-fluorophenyl)-1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}ethan-1-one
2-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}-2-[4-(1H-pyrazol-5-yl)phenyl]acetic acid
4-(5-benzyl-2-methylpyrimidin-4-yl)-N,N-dimethylpiperidine-1-sulfonamide
4-(4-chlorophenoxy)-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidine
2,6-dimethyl-5-{2-oxo-2-[4-(9H-purin-6-yl)piperazin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[4-(pyridin-2-yl)butyl]pyridin-2-amine
5-(2H-1,3-benzodioxol-4-yl)-1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazole
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(4-methylphenyl)piperazine
1-(furan-2-carbonyl)-3-[4-phenyl-5-(propan-2-yl)-1H-imidazol-1-yl]piperidine
8-(1H-indol-3-ylmethyl)-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-methyl-5-{5-[1-(pyrimidin-2-yl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
1-ethyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
1-(4-benzylpiperazine-1-carbonyl)-6-[(4-methoxy-3-methylphenyl)methyl]-6-azaspiro[2.5]octane
N3-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-N1-(pyridin-3-yl)propane-1,3-diamine
(2R,6R)-4-{[3-(2-hydroxyethoxy)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-({[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)amino}methyl)-6,7-dimethyl-2H-chromen-2-one
N-[2-(ethylsulfanyl)ethyl]-4-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}benzamide
4-{1-[(2,5-difluorophenyl)methyl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
methyl 2-(3-oxo-4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-2-yl)acetate
3-{1-[2-(3-chlorophenyl)acetyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
1-[2-(dimethylamino)-4-{[2-(phenylamino)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one