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7-cyclopentyl-2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-3-(1H-pyrazol-1-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
2-(4-chlorophenyl)-N-[2-(3-methylpyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-(adamantan-1-ylmethyl)-2-[1-(2-methoxyethyl)-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
N-[2-(4-fluorophenyl)ethyl]-N-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-chloro-N-[2-(1,3-thiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
7-(hydroxymethyl)-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
methyl 3-[(2,5-dimethoxyphenyl)methyl]-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidine-3-carboxylic acid
5-benzyl-4-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-3-yl}-2-methylpyrimidine
4-(4-chlorophenyl)-1-[4-(cyclobutylmethyl)piperazin-1-yl]butan-1-one
2-[(5-methylpyrazin-2-yl)methyl]-9-(5-methylthiophene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
3-methyl-5-(oxan-4-yl)-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
5-[1-methyl-5-(trifluoromethyl)-1H-pyrazole-3-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)[(4-methylphenyl)methyl]amine
N-(1-{1-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(thiophene-2-carbonyl)piperidine
6-methoxy-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyrimidin-4-amine
2,3,6-trimethyl-4-[4-(pyridin-4-yl)piperidine-1-carbonyl]quinoline
2-[(2-chlorophenyl)methyl]-4-[4-(2-methylpropyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-oxazepane
4-(5-{[4-(pentan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-1,2,4-triazol-3-yl)pyridine
1,3-dimethyl-6-{6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-benzyl-N-methyl-2-{[(oxolan-3-ylmethyl)amino]methyl}-2,3-dihydro-1H-inden-2-amine
2,6-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-3-carboxamide
6-ethyl-4-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)-2H-chromen-2-one
ethyl 1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
N-{3-[4-(acetamidomethyl)-5-methyl-1,3-oxazol-2-yl]phenyl}-2-(4-methylphenoxy)acetamide
3-{4-[(4-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}-1,2-benzothiazole
6-methoxy-N-[4-(morpholin-4-ylmethyl)phenyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]-2-(morpholin-4-yl)propan-1-one
3-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
5-(2,4-difluorophenoxymethyl)-3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazole
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methanol
4-(dimethyl-1,2-oxazol-4-yl)-3-(3,4,5-trimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,4-dimethoxybenzamide
(3aS,7aR)-2-[(5-chlorothiophen-2-yl)methyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
5-(2-chlorophenyl)-2-methyl-N-(pyridin-4-ylmethyl)furan-3-carboxamide
N5-[2-(cyclohex-1-en-1-yl)ethyl]-N3,N3-diethyl-1-[(2-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
({3-[(4-ethylpiperazin-1-yl)methyl]-2,5-dimethylphenyl}methyl)(methyl)(pyridin-2-ylmethyl)amine
N-(2-ethoxybutyl)-5-fluoro-1,3-dimethyl-1H-indole-2-carboxamide
N-(3,3-diphenylpropyl)-6-[(5-methylfuran-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
6-ethoxy-2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1,4-diazepan-1-yl}-4-methylquinazoline
N-[(3,4-dimethoxyphenyl)methyl]-2,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-indole-7-carboxamide